CAS 2913231-72-6

Glucocorticoid receptor agonist-5

Description:

Glucocorticoid receptor agonist-5, identified by its CAS number 2913231-72-6, is a synthetic compound that acts as an agonist for the glucocorticoid receptor (GR). This receptor is a type of nuclear receptor that, upon binding with glucocorticoids, regulates the expression of various genes involved in inflammation, immune response, and metabolism. Compounds like glucocorticoid receptor agonist-5 are typically characterized by their ability to modulate GR activity, potentially leading to anti-inflammatory and immunosuppressive effects. These properties make them of interest in therapeutic applications for conditions such as autoimmune diseases, allergies, and certain inflammatory disorders. The pharmacokinetics, potency, and selectivity of this compound can vary, influencing its efficacy and safety profile. Additionally, the development of such agonists often aims to minimize side effects commonly associated with traditional glucocorticoids, such as metabolic disturbances and adrenal suppression. Further research is essential to fully understand the biological effects and therapeutic potential of glucocorticoid receptor agonist-5.

Formula: C₃₆H₄₀O₇

Synonyms:

• Pregna-1,4-diene-3,20-dione, 11,21-dihydroxy-16,17-[[(R)-[4-[[4-(hydroxymethyl)phenyl]methyl]phenyl]methylene]bis(oxy)]-, (11β,16α)-
• Glucocorticoid receptor agonist-5

Glucocorticoid receptor agonist-5

CAS: 2913231-72-6

Glucocorticoid Receptoragonist-5 (compound 4) is an effective glucocorticoid molecule acting as a potent agonist for glucocorticoid receptors. It exhibits anti-inflammatory and immunosuppressive activities and serves as an ADC cytotoxin.

Formula: C₃₆H₄₀O₇

Color and Shape: Solid

Molecular weight: 584.7

Ref: TM-T201729