CAS 30123-17-2

Tianeptine sodium

Description:

Tianeptine sodium, with the CAS number 30123-17-2, is the sodium salt form of tianeptine, a compound primarily known for its antidepressant properties. It is classified as a selective serotonin reuptake enhancer (SSRE), which distinguishes it from traditional SSRIs that inhibit serotonin reuptake. Tianeptine sodium is typically presented as a white to off-white crystalline powder, soluble in water, which facilitates its use in various formulations. The compound is known to influence the glutamatergic system and has neuroprotective effects, making it of interest in the treatment of mood disorders and anxiety. Additionally, tianeptine sodium has been studied for its potential benefits in cognitive function and stress resilience. Its pharmacokinetics involve rapid absorption and a relatively short half-life, necessitating careful dosing. While it is not approved for use in some countries, it remains a subject of research and discussion in the context of mental health treatment. As with any pharmacological agent, understanding its safety profile and potential side effects is crucial for its therapeutic application.

Formula: C₂₁H₂₅ClN₂O₄S·Na

InChI: InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);

InChI key: InChIKey=UDFCCNYPCCUJOO-UHFFFAOYSA-N

SMILES: N(CCCCCCC(O)=O)C1C=2C(S(=O)(=O)N(C)C=3C1=CC=CC3)=CC(Cl)=CC2.[Na]

Synonyms:

• Dibenzo[c,f][1,2]thiazepine, heptanoic acid deriv.
• Heptanoic acid, 7-[(3-chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]-, monosodium salt
• Heptanoic acid, 7-[(3-chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]-, sodium salt (1:1)
• Heptanoic acid, 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]-, S,S-dioxide, monosodium salt
• Sodium 7-[(3-chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoate
• Stablon
• Tianeptine Sodium
• Tianeptine sodium salt
• [7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepine 5,5-dioxide)-11-ylamino]heptanoic acid]sodium salt

Tianeptine Sodium Salt

CAS: 30123-17-2, 72797-41-2

Formula: C₂₁H₂₄ClN₂NaO₄S

Purity: >98.0%(HPLC)(N)

Color and Shape: White to Almost white powder to crystal

Molecular weight: 458.93

Ref: 3B-T3131

SODIUM TIANEPTINE FOR SYSTEM SUITABILITY CRS

CAS: 30123-17-2

SODIUM TIANEPTINE FOR SYSTEM SUITABILITY CRS

Formula: C₈H₁₆O₂

Molecular weight: 144.2114

Ref: 41-Y0000152

Tianeptine (sodium salt)

CAS: 30123-17-2

Formula: C₂₁H₂₄ClN₂NaO₄S

Purity: 98%

Color and Shape: Solid

Molecular weight: 458.9340

Ref: IN-DA0037EM

Tianeptine Sodium Salt

CAS: 30123-17-2

Formula: C₂₁H₂₄ClN₂O₄S·Na

Color and Shape: White To Off-White Solid

Molecular weight: 435.95 22.99

Ref: 4Z-T-361

Tianeptine Sodium

CAS: 30123-17-2

Formula: C₂₁H₂₄ClN₂O₄S·Na

Color and Shape: Neat

Molecular weight: 458.93

Ref: 86-MM3456.00

Tianeptine sodium salt

CAS: 30123-17-2

Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。

Formula: C₂₁H₂₄ClN₂NaO₄S

Purity: 99.82%

Color and Shape: Solid

Molecular weight: 458.93

Ref: TM-T2402

Tianeptine sodium salt hydrate

CAS: 30123-17-2

Formula: C₂₁H₂₄ClN₂NaO₄S·xH₂O

Purity: ≥ 98.0%

Color and Shape: White to off-white powder

Molecular weight: 458.93

Ref: 7W-GP8667

Tianeptine-d12

CAS: 30123-17-2

Formula: C₂₁H₁₃ClN₂O₄SD₁₂

Molecular weight: 448.95 22.99

Ref: 4Z-T-362

Tianeptine Sodium Salt

CAS: 30123-17-2

Applications Tianeptine Sodium Salt is a tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant.
References Malen, C., et al.: Experientia, 28, 811 (1972),

Formula: C₂₁H₂₄ClN₂O₄S·Na

Color and Shape: Off-White

Molecular weight: 458.93

Ref: TR-T436805

Tianeptine sodium salt - Bio-X ™

Controlled Product

CAS: 30123-17-2

Tianeptine is a tricyclic antidepressant with anxiolytic effects to treat major depressive disorder. Additionally, this drug has been studied for the treatment of irritable bowel syndrome. Studies have suggested that this drug is an agonist of the mu-type opioid receptor. This drug also exerts its action on serotonin and dopamine receptors.

Formula: C₂₁H₂₅ClN₂O₄S•Na

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 459.93 g/mol

Ref: 3D-BT164468

Tianeptine sodium salt

Controlled Product

CAS: 30123-17-2

Full agonist of the μ-opioid receptor (MOR) with Ki of 383 nM. It also weakly agonizes the δ-opioid receptor (DOR) with a Ki >10 μM. Tianeptine has antidepressant effects but can also regulate neuroplasticity in the amygdala and stress-induced release of glutamate. It can generate analgesia and reward, typical opiate-like behavioural effects, but does not induce tolerance or withdrawal.

Formula: C₂₁H₂₄ClN₂NaO₄S

Purity: Min. 98.5 Area-%

Color and Shape: White Slightly Yellow Powder

Molecular weight: 458.93 g/mol

Ref: 3D-FT28266