CAS 313-06-4

Estradiol cypionate

Description:

Estradiol cypionate is a synthetic form of the naturally occurring estrogen estradiol, classified as a steroid hormone. It is primarily used in hormone replacement therapy and for various medical conditions related to estrogen deficiency. The substance is characterized by its chemical structure, which includes a cypionate ester that enhances its solubility and prolongs its action in the body. Estradiol cypionate is typically administered via intramuscular injection, allowing for gradual release into the bloodstream. Its pharmacological effects include the regulation of the menstrual cycle, alleviation of menopausal symptoms, and support of bone density. The compound is known for its relatively high potency and efficacy in promoting estrogenic activity. Common side effects may include headaches, mood changes, and potential cardiovascular risks, necessitating careful monitoring during treatment. As with all hormonal therapies, the use of estradiol cypionate should be tailored to individual patient needs and medical history, ensuring a balance between therapeutic benefits and potential risks.

Formula: C₂₆H₃₆O₃

InChI: InChI=1S/C26H36O3/c1-26-15-14-21-20-10-8-19(27)16-18(20)7-9-22(21)23(26)11-12-24(26)29-25(28)13-6-17-4-2-3-5-17/h8,10,16-17,21-24,27H,2-7,9,11-15H2,1H3/t21-,22-,23+,24+,26+/m1/s1

InChI key: InChIKey=UOACKFBJUYNSLK-XRKIENNPSA-N

SMILES: C[C@@]12[C@]([C@]3([C@@](C=4C(CC3)=CC(O)=CC4)(CC1)[H])[H])(CC[C@@H]2OC(CCC5CCCC5)=O)[H]

Synonyms:

• (17Beta)-3-Hydroxyestra-1,3,5(10)-Trien-17-Yl 3-Cyclopentylpropanoate
• (8Xi,9Xi,14Xi,17Beta)-3-Hydroxyestra-1,3,5(10)-Trien-17-Yl 3-Cyclopentylpropanoate
• 17β-Estradiol 17-cyclopentylpropionate
• 3-Hydroxyestra-1,3,5(10)-Trien-17-Yl 3-Cyclopentylpropanoate
• Cyclopentanepropionic acid, 17-ester with estradiol
• Cyclopentanepropionic acid, 3-hydroxyestra-1,3,5(10)-trien-17β-yl ester
• Depgynogen
• Depo-Estradiol
• Depo-estradiol cyclopentylpropionate
• Depoestradiol
• Depoestradiol cypionate
• Depofemin
• Estra-1,3,5(10)-triene-3,17-diol (17β)-, 17-cyclopentanepropanoate
• Estradep
• Estradiol 17-Beta-(3-Cyclopentylpropionate)
• Estradiol 17-Beta-Cipionate
• Estradiol 17-Cypionate
• Estradiol 17-cyclopentylpropionate
• Estradiol 17β-cyclopentanepropionate
• Estradiol 17β-cyclopentylpropionate
• Estradiol 17β-cypionate
• Estradiol Cypionate
• Estradiol cyclopentylpropionate
• Estradiol, 17-cyclopentanepropionate
• Estradiolum valerianicum
• NSC 3354

Estradiol Cypionate

CAS: 313-06-4

Color and Shape: Neat

Ref: 61-FOR3402.00

Estradiol Cypionate

CAS: 313-06-4

Estrogens and progestins

Formula: C₂₆H₃₆O₃

Color and Shape: White Off-White Powder

Molecular weight: 396.26645

Ref: 45-1252003

Estradiol (cypionate)

CAS: 313-06-4

Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor.

Formula: C₂₆H₃₆O₃

Purity: 99.53% - >99.99%

Color and Shape: White Or Off-White Crystalline Powder

Molecular weight: 396.56

Ref: TM-T0168

β-Estradiol 17-Cypionate

CAS: 313-06-4

β-Estradiol 17-Cypionate

Purity: 99%

Molecular weight: 396.56g/mol

Ref: 54-OR1028757

Estradiol (cypionate)

CAS: 313-06-4

Estradiol (cypionate)

Purity: ≥98%

Molecular weight: 396.56g/mol

Ref: 54-BUP17759

Estradiol cypionate

CAS: 313-06-4

Formula: C₂₆H₃₆O₃

Molecular weight: 396.56

Ref: 7W-GP8937

Estradiol Cypionate

Controlled Product

CAS: 313-06-4

Formula: C₂₆H₃₆O₃

Color and Shape: Neat

Molecular weight: 396.56

Ref: 86-MM3402.00

17-β-Estradiol 17-cypionate

CAS: 313-06-4

Color and Shape: Neat

Ref: 04-C13213125

Estradiol Cypionate

CAS: 313-06-4

Applications Estradiol Cypionate is present in injectable contraceptive formulations. Used in hormone replacement therapy with potential for improving cognition in post-menopausal women.
References Thurman, A. et al.: Contra., 87, 738 (2013); Sales, J. et al.: Theriogen., 78, 510 (2012); Rapp, P. et al.: J. neurosci., 23, 5708 (2003);

Formula: C₂₆H₃₆O₃

Color and Shape: Neat

Molecular weight: 396.56

Ref: TR-E668610

Estradiol cypionate

CAS: 313-06-4

Estradiol cypionate is a synthetic form of estrogen. It is used as a contraceptive and to treat certain types of breast cancer. Estradiol cypionate is administered by intramuscular injection, and has been shown to be effective in inhibiting ovulation, ovarian activity, and follicular growth. Estradiol cypionate is metabolized in the liver to estradiol benzoate and estrone, which have similar effects on the body. The pharmacokinetics of estradiol cypionate are complex because it binds to sex hormone-binding globulin (SHBG) in the blood serum. This binding reduces the availability of free estradiol for receptor binding, which may result in decreased effectiveness with long-term use.

Formula: C₂₆H₃₆O₃

Purity: Min. 95%

Color and Shape: White Powder

Molecular weight: 396.56 g/mol

Ref: 3D-FE61563