CAS 34661-85-3

5-Methylurapidil

Description:

5-Methylurapidil is a chemical compound that belongs to the class of selective alpha-1 adrenergic antagonists, primarily used in the treatment of hypertension. It is characterized by its ability to selectively block alpha-1 adrenergic receptors, leading to vasodilation and a subsequent decrease in blood pressure. The molecular structure of 5-Methylurapidil includes a methyl group at the 5-position of the urapidil framework, which contributes to its pharmacological properties. This compound exhibits moderate solubility in water and is typically administered in oral form. Its mechanism of action not only involves alpha-1 receptor antagonism but also includes central effects that may influence blood pressure regulation. Additionally, 5-Methylurapidil has been studied for its potential effects on other cardiovascular parameters and may have implications in treating conditions beyond hypertension. As with any pharmaceutical agent, its use should be guided by clinical considerations and potential side effects.

Formula: C₂₁H₃₁N₅O₃

InChI: InChI=1S/C21H31N5O3/c1-16-19(23(2)21(28)24(3)20(16)27)22-10-7-11-25-12-14-26(15-13-25)17-8-5-6-9-18(17)29-4/h5-6,8-9,22H,7,10-15H2,1-4H3

InChI key: InChIKey=HIHZDNKKIUQQSC-UHFFFAOYSA-N

SMILES: O(C)C1=C(C=CC=C1)N2CCN(CCCNC3=C(C)C(=O)N(C)C(=O)N3C)CC2

Synonyms:

• 2,4(1H,3H)-pyrimidinedione, 6-[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3,5-trimethyl-
• 5-Methylurapidil
• 5-Methyluropidil
• 6-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3,5-trimethyl-2,4(1H,3H)-pyrimidinedione
• 6-({3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}amino)-1,3,5-trimethylpyrimidine-2,4(1H,3H)-dione

5-Methylurapidil

CAS: 34661-85-3

Formula: C₂₁H₃₁N₅O₃

Molecular weight: 401.50

Ref: 7W-GL2645

5-Methylurapidil

CAS: 34661-85-3

Formula: C₂₁H₃₁N₅O₃

Molecular weight: 401.51

Ref: 4Z-U-0720

5-Methylurapidil

Controlled Product

CAS: 34661-85-3

Formula: C₂₁H₃₁N₅O₃

Color and Shape: Neat

Molecular weight: 401.502

Ref: TR-M338178

5-Methylurapidil

CAS: 34661-85-3

5-Methylurapidil is an alpha1A-adrenoceptor antagonist.

Formula: C₂₁H₃₁N₅O₃

Purity: 98%

Color and Shape: Solid

Molecular weight: 401.5

Ref: TM-T26393