CAS 3505-38-2

carbinoxamine maleate

Description:

Carbinoxamine maleate is an antihistamine used primarily for the relief of allergy symptoms, such as hay fever and other allergic conditions. It functions as a first-generation H1 receptor antagonist, which means it blocks the action of histamine, a substance in the body that causes allergic symptoms. The compound is typically administered in the form of its maleate salt, enhancing its solubility and stability. Carbinoxamine maleate is characterized by its ability to cross the blood-brain barrier, which can lead to sedative effects, a common trait of first-generation antihistamines. It is often used in combination with other medications to treat cold symptoms and is available in various formulations, including tablets and syrups. The substance has a relatively low toxicity profile when used as directed, but potential side effects may include drowsiness, dry mouth, and dizziness. As with any medication, it is essential to use carbinoxamine maleate under the guidance of a healthcare professional to ensure safety and efficacy.

Formula: C₂₀H₂₃ClN₂O₅

InChI: InChI=1/C16H19ClN2O.C4H4O4/c1-19(2)11-12-20-16(15-5-3-4-10-18-15)13-6-8-14(17)9-7-13;5-3(6)1-2-4(7)8/h3-10,16H,11-12H2,1-2H3;1-2H,(H,5,6)(H,7,8)/p-2/b;2-1-

InChI key: InChIKey=GVNWHCVWDRNXAZ-BTJKTKAUSA-N

SMILES: C(OCCN(C)C)(C1=CC=C(Cl)C=C1)C2=CC=CC=N2.C(=C\C(O)=O)\C(O)=O

Synonyms:

• 2-[(4-chlorophenyl)(pyridin-2-yl)methoxy]-N,N-dimethylethanamine
• 2-[(4-chlorophenyl)(pyridin-2-yl)methoxy]-N,N-dimethylethanamine (2Z)-but-2-enedioate
• 2-[p-Chloro-α-[2-(dimethylamino)ethoxy]benzyl]pyridine Bimaleate
• 2-[p-Chloro-α-[2-(dimethylamino)ethoxy]benzyl]pyridine maleate
• Allergefon
• Allergefon maleate
• Carbinoxamine Hydrogen Maleate
• Carbinoxamine Maleate Salt
• Ciberon
• Clistin
• Clistine Maleate
• Cliston
• Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-, (2Z)-2-butenedioate (1:1)
• Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-, (Z)-2-butenedioate (1:1)
• Hislosine
• Lergefin
• NSC 62362
• Paracarbinoxamine maleate
• Polistin T-Caps
• Pyridine, 2-[p-chloro-α-[2-(dimethylamino)ethoxy]benzyl]-, maleate (1:1)
• Rondec
• Rondec DM
• Carbinoxamine maleate
• 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-n,n-dimethyl-ethanamin(z)-2-butene
• clistinemaleate
• 2-(p-chloro-alpha-(2-(dimethylamino)ethoxy)benzyl)pyridinebimaleate
• 2-(p-chloro-alpha-(2-(dimethylamino)ethoxy)benzyl)pyridinemaleate
• allergefonmaleate
• 2-(p-chloro-alpha-(2-(dimethylamino)ethoxy)benzyl)-pyridinmaleate(1:1)
• 2-((4-chlorophenyl)-2-pyridinylmethoxy)-n,n-dimethyl-ethanamin(z)-2-bute
• p-carbinoxaminemaleate
• 2-[(4-Clorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-ethanamine Maleate Salt
• clistinmaleate

Carbinoxamine Maleate

CAS: 3505-38-2, 486-16-8

Formula: C₁₆H₁₉ClN₂O·C₄H₄O₄

Purity: >98.0%(T)(HPLC)

Color and Shape: White to Almost white powder to crystal

Molecular weight: 406.86

Ref: 3B-C3057

Carbinoxamine Maleate

CAS: 3505-38-2

Color and Shape: Neat

Ref: 61-FOR1135.00

Carbinoxamine Maleate

CAS: 3505-38-2

Compounds containing an unfused pyridine ring in the structure, nesoi

Formula: C₁₆H₁₉ClN₂O·C₄H₄O₄

Color and Shape: White Crystalline Powder

Molecular weight: 406.12955

Ref: 45-1096000

Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-,(2Z)-2-butenedioate (1:1)

CAS: 3505-38-2

Formula: C₂₀H₂₃ClN₂O₅

Purity: %

Color and Shape: Solid

Molecular weight: 406.8600

Ref: IN-DA00I6XV

Carbinoxamine Maleate Salt

CAS: 3505-38-2

Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.

Formula: C₂₀H₂₃ClN₂O₅

Purity: 99.97%

Color and Shape: Off-White Solid

Molecular weight: 406.86

Ref: TM-T2222

Carbinoxamine Maleate

CAS: 3505-38-2

Formula: C₁₆H₁₉ClN₂O·C₄H₄O₄

Color and Shape: White To Off-White Solid

Molecular weight: 290.80 116.07

Ref: 4Z-C-672

Carbinoxamine Maleate Salt

CAS: 3505-38-2

Carbinoxamine Maleate Salt

Purity: ≥98%

Molecular weight: 406.86g/mol

Ref: 54-BUP15772

Carbinoxamine Maleate

CAS: 3505-38-2

Carbinoxamine Maleate

Purity: 99%

Molecular weight: 406.86g/mol

Ref: 54-OR1028594

Carbinoxamine maleate salt

CAS: 3505-38-2

Formula: C₁₆H₁₉ClN₂O·C₄H₄O₄

Purity: 99.0 - 101.0 % (dried basis)

Color and Shape: White to almost white powder

Molecular weight: 406.86

Ref: 7W-GP7553

Carbinoxamine-d6 Maleate

CAS: 3505-38-2

Formula: C₁₆H₁₃D₆ClN₂O·C₄H₄O₄

Color and Shape: Off-White Solid

Molecular weight: 296.83 116.07

Ref: 4Z-C-671

(±)-Carbinoxamide-d6 Maleate(N,N-dimethyl-d6)

CAS: 3505-38-2

Purity: 98 atom % D

Color and Shape: White Solid

Molecular weight: 412.90

Ref: 3U-D7564

Carbinoxamine Maleate

CAS: 3505-38-2

Color and Shape: Neat

Ref: 86-MM1135.00

Carbinoxamine Maleate Salt

Controlled Product

CAS: 3505-38-2

Applications Analgesic and anti-inflammatory compound.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Cochin, J., et al.: J. Pharmacol. Exp. Ther., 139, 160 (1963),

Formula: C₁₆H₁₉ClN₂O·C₄H₄O₄

Color and Shape: Neat

Molecular weight: 406.86

Ref: TR-C175920

2-[(4-Chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethylethanamine maleate salt

Controlled Product

CAS: 3505-38-2

2-[(4-Chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethylethanamine maleate salt (DCLM) is a controlled-release preparation of an antihistamine that is used for the relief of allergic symptoms. It is a prodrug that is hydrolyzed to 2-[(4-chlorophenyl)-2-pyridinylmethoxy]ethanol (DCPEM) in vivo. DCLM has been shown to be effective against viruses and has been found to have receptor activity in human serum. The drug can be administered either orally or by injection. DCLM has also been shown to suppress allergic symptoms in vitro with LC-MS/MS analysis.

Formula: C₂₀H₂₃ClN₂O₅

Purity: Min. 95%

Color and Shape: White To Off-White Solid

Molecular weight: 406.86 g/mol

Ref: 3D-FC19699

Carbinoxamine maleate

CAS: 3505-38-2

Purity: 98%

Molecular weight: 406.86

Ref: 10-F825776