CAS 3505-38-2: carbinoxamine maleate
Description:Carbinoxamine maleate is an antihistamine used primarily for the relief of allergy symptoms, such as hay fever and other allergic conditions. It functions as a first-generation H1 receptor antagonist, which means it blocks the action of histamine, a substance in the body that causes allergic symptoms. The compound is typically administered in the form of its maleate salt, enhancing its solubility and stability. Carbinoxamine maleate is characterized by its ability to cross the blood-brain barrier, which can lead to sedative effects, a common trait of first-generation antihistamines. It is often used in combination with other medications to treat cold symptoms and is available in various formulations, including tablets and syrups. The substance has a relatively low toxicity profile when used as directed, but potential side effects may include drowsiness, dry mouth, and dizziness. As with any medication, it is essential to use carbinoxamine maleate under the guidance of a healthcare professional to ensure safety and efficacy.
Formula:C20H21ClN2O5
InChI:InChI=1S/C16H19ClN2O.C4H4O4/c1-19(2)11-12-20-16(15-5-3-4-10-18-15)13-6-8-14(17)9-7-13;5-3(6)1-2-4(7)8/h3-10,16H,11-12H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
InChI key:InChIKey=GVNWHCVWDRNXAZ-BTJKTKAUSA-N
SMILES:O=C(O)C=CC(=O)O.ClC1=CC=C(C=C1)C(OCCN(C)C)C2=NC=CC=C2
- Synonyms:
- 2-[(4-chlorophenyl)(pyridin-2-yl)methoxy]-N,N-dimethylethanamine
- 2-[(4-chlorophenyl)(pyridin-2-yl)methoxy]-N,N-dimethylethanamine (2Z)-but-2-enedioate
- 2-[p-Chloro-α-[2-(dimethylamino)ethoxy]benzyl]pyridine Bimaleate
- 2-[p-Chloro-α-[2-(dimethylamino)ethoxy]benzyl]pyridine maleate
- Allergefon
- Allergefon maleate
- Carbinoxamine Hydrogen Maleate
- Carbinoxamine Maleate Salt
- Ciberon
- Clistin
- See more synonyms
- Clistine Maleate
- Cliston
- Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-, (2Z)-2-butenedioate (1:1)
- Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-, (Z)-2-butenedioate (1:1)
- Hislosine
- Lergefin
- NSC 62362
- Paracarbinoxamine maleate
- Polistin T-Caps
- Pyridine, 2-[p-chloro-α-[2-(dimethylamino)ethoxy]benzyl]-, maleate (1:1)
- Rondec
- Rondec DM