CAS 359-83-1

Pentazocine

Description:

Pentazocine is a synthetic opioid analgesic primarily used for the relief of moderate to severe pain. It is classified as a mixed agonist-antagonist, meaning it can activate certain opioid receptors while simultaneously blocking others, which can reduce the risk of dependence compared to pure agonists. Pentazocine has a complex chemical structure, characterized by a bicyclic system that contributes to its pharmacological properties. It is typically administered via oral or parenteral routes and has a relatively rapid onset of action. The substance is known to produce effects such as analgesia, sedation, and euphoria, but it may also lead to side effects including dizziness, nausea, and potential respiratory depression. Due to its potential for abuse and dependence, pentazocine is classified as a controlled substance in many jurisdictions. Its use is often limited to specific clinical scenarios, and it is important for healthcare providers to monitor patients closely for signs of misuse or adverse reactions.

Formula: C₁₉H₂₇NO

InChI: InChI=1/C19H27NO/c1-13(2)7-9-20-10-8-19(4)14(3)18(20)11-15-5-6-16(21)12-17(15)19/h5-7,12,14,18,21H,8-11H2,1-4H3/t14-,18+,19+/s2

InChI key: InChIKey=VOKSWYLNZZRQPF-RWKILVNUNA-N

SMILES: C[C@@]12C=3C(C[C@@]([C@H]1C)(N(CC=C(C)C)CC2)[H])=CC=C(O)C3

Synonyms:

• (.+-.)-Pentazocine
• 1,2,3,4,5,6-Hexahydro-3-(3-methyl-2-butenyl)-6,11-dimethyl-8-hydroxy-2,6-methano-3-benzazocine
• 1,2,3,4,5,6-Hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocin-8-ol
• 2'-Hydroxy-5,9-dimethyl-2-(3,3-dimethylallyl)-6,7-benzomorphan
• 2,6-Methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-buten-1-yl)-, (2R,6R,11R)-rel-
• 2,6-Methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-, (2α,6α,11R*)-
• 2-Dimethylallyl-5,9-dimethyl-2'-hydroxybenzomorphan
• 3-(3-Methyl-2-butenyl)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-2,6-methano-3-benzazocin-8-ol
• 3-(3-Methyl-2-butenyl)-1,2,3,4,5,6-hexahydro-8-hydroxy-6,11-dimethyl-2,6-methano-3-benzazocine
• Fortalgesic
• Fortalin
• Fortral
• Fortwin
• Ii-C 2
• Lexir
• Nih 7958
• Nsc 107430
• Peltazon
• Pentagin
• Pentazocin
• Pentazocina
• Pentazocine Usp Recrystallized
• Sosegon
• Soseton
• Sosigon
• Talwin
• Win 20228
• cis-(.+-.)-Pentazocine
• dl-Pentazocine
• rel-(2R,6R,11R)-1,2,3,4,5,6-Hexahydro-6,11-dimethyl-3-(3-methyl-2-buten-1-yl)-2,6-methano-3-benzazocin-8-ol

Pentazocine

Controlled Product

CAS: 359-83-1

Applications Mixed opioid agonist-antagonist. Controlled substance. Analgesic (narcotic).
References Goldenthal, E.I., et al.: Toxicol. Appl. Pharmacol., 18, 185 (1971), Brogden, et al.: Drugs, 5, 6 (1973), Camu, F., et al.: Eur. J. Clin. Pharmacol., 19, 259 (1981),

Formula: C₁₉H₂₇NO

Color and Shape: Beige To Light Brown

Molecular weight: 285.42

Ref: TR-P274300

Pentazocine (1 mg/ml in Methanol)

Controlled Product

CAS: 359-83-1

Formula: C₁₉H₂₇NO

Color and Shape: Colourless

Molecular weight: 285.42

Ref: TR-KIT2375

Pentazocine CIV

Controlled Product

CAS: 359-83-1

Alfentanil (inn), anileridine (inn), bezitramide (inn), bromazepam (inn), difenoxin (inn), diphenoxylate (inn), dipipanone (inn), fentanyl (inn), etc.

Formula: C₁₉H₂₇NO

Color and Shape: White Beige Crystalline Powder

Molecular weight: 285.43

Ref: 45-1505007

Pentazocine

Controlled Product

CAS: 359-83-1

Pentazocine is a nonsteroidal anti-inflammatory drug that is used to relieve pain. It has been shown to bind to the kappa-opioid receptor, which may be responsible for pentazocine's analgesic effects. Pentazocine also has a low potency and side-effect profile, as well as some physiological effects such as respiratory depression. Pentazocine is not active in the central nervous system and can be administered by nasal route. The drug has been shown to have an additive effect when combined with isoxsuprine hydrochloride in patients with eosinophilic fasciitis. Pentazocine is also used as a pharmacological treatment for myocardial infarcts and other cardiovascular disorders.

Formula: C₁₉H₂₇NO

Purity: Min. 95%

Molecular weight: 285.42 g/mol

Ref: 3D-FP26819