CAS 3900-31-0

Fludiazepam

Description:

Fludiazepam is a benzodiazepine derivative known for its anxiolytic, sedative, and muscle relaxant properties. It is characterized by its ability to enhance the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased neuronal inhibition. This compound typically exhibits a rapid onset of action and a relatively long duration of effects, making it useful in clinical settings for managing anxiety and sleep disorders. Fludiazepam is often administered in the form of oral tablets, and its pharmacokinetics can vary based on individual metabolism and dosage. Common side effects may include drowsiness, dizziness, and potential dependence with prolonged use. Due to its psychoactive properties, fludiazepam is classified as a controlled substance in many jurisdictions, necessitating careful regulation and monitoring in medical use. As with other benzodiazepines, caution is advised when prescribing fludiazepam, particularly in patients with a history of substance abuse or those taking other central nervous system depressants.

Formula: C₁₆H₁₂ClFN₂O

InChI: InChI=1S/C16H12ClFN2O/c1-20-14-7-6-10(17)8-12(14)16(19-9-15(20)21)11-4-2-3-5-13(11)18/h2-8H,9H2,1H3

InChI key: InChIKey=ROYOYTLGDLIGBX-UHFFFAOYSA-N

SMILES: FC1=C(C=2C=3C(N(C)C(=O)CN2)=CC=C(Cl)C3)C=CC=C1

Synonyms:

• 2H-1,4-Benzodiazepin-2-one, 7-chloro-5-(o-fluorophenyl)-1,3-dihydro-1-methyl-
• 7-Chloro-5-(2-fluorophenyl)-1,3-dihydro-1-methyl-2H-1,4-benzodiazepin-2-one
• 7-Chloro-5-(2-fluorophenyl)-1-methyl-1,3-dihydrobenzo[e][1,4]diazepin-2-one
• 7-Chloro-5-(2-fluorophenyl)-1-methyl-1H-1,4-benzodiazepin-2(3H)-one
• Erispan
• Fludiazepam
• Id 540
• Ro 5-3438
• Fludiazepamum [INN-Latin]
• Fludiazepam [INN:JAN]
• DEA No. 2759
• UNII-7F64A2K16Z
• 5-24-04-00320 (Beilstein Handbook Reference)
• Fludiazepamum
• 2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-7-chloro-5-(o-fluorophenyl)-1-methyl-
• 7-Chloro-5-(o-Fluorophenyl)-1,3-dihydro-1-methyl-2H-1,4-benzodiazepin-2-one
• 2H-1,4-Benzodiazepin-2-one, 7-chloro-5-(2-fluorophenyl)-1,3-dihydro-1-methyl-
• BRN 0686115
• 2H-1,4-Benzodiazepin-2-one, 7-chloro-5-(2-fluorophenyl)-1,3-dihydro-1-methyl- (9CI)

Fludiazepam, 1mg/ml in Methanol

Controlled Product

CAS: 3900-31-0

Color and Shape: Single Solution

Ref: LP-FLD-396-1LM

Fludiazepam

Controlled Product

CAS: 3900-31-0

Color and Shape: Neat

Ref: LP-FLD-396-10

Fludiazepam

Controlled Product

CAS: 3900-31-0

Applications Fludiazepam is a drug which is a benzodiazepine derivative. Fludiazepam possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties.
References Fang, S.Y., et al.: Drug. Alcohol. Depend., 104, 140 (2009); Esteki, M., et al.: Chem. Biol. Drug. Design., 72, 409 (2008);

Formula: C₁₆H₁₂ClFN₂O

Color and Shape: White To Off-White

Molecular weight: 302.7307

Ref: TR-F428800

Fludiazepam-d3

Controlled Product

CAS: 3900-31-0

Applications Isotope Labelled Fludiazepam is a drug which is a benzodiazepine derivative. Fludiazepam possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties.
References Fang, S.Y., et al.: Drug. Alcohol. Depend., 104, 140 (2009); Esteki, M., et al.: Chem. Biol. Drug. Design., 72, 409 (2008);

Formula: C₁₆D₃H₉ClFN₂O

Color and Shape: Neat

Molecular weight: 305.749

Ref: TR-F428802