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CAS 42281-59-4

:

Oxilorphan

Description:
Oxilorphan is a synthetic compound primarily recognized for its role as an opioid receptor antagonist, particularly at the mu-opioid receptor, while also exhibiting some agonistic properties at the kappa-opioid receptor. Its chemical structure includes a phenolic hydroxyl group, which contributes to its pharmacological activity. Oxilorphan is often studied for its potential applications in pain management and as a treatment for opioid dependence, as it can mitigate the effects of opioid overdose. The substance is characterized by its ability to cross the blood-brain barrier, influencing central nervous system activity. Additionally, it has been investigated for its neuroprotective properties and potential use in various neurological conditions. However, its clinical use is limited, and it is primarily of interest in research settings. As with many compounds that interact with opioid receptors, careful consideration of its pharmacodynamics and potential side effects is essential in any therapeutic context.
Formula:C20H27NO2
InChI:InChI=1S/C20H27NO2/c22-16-6-5-15-11-18-20(23)8-2-1-7-19(20,17(15)12-16)9-10-21(18)13-14-3-4-14/h5-6,12,14,18,22-23H,1-4,7-11,13H2/t18-,19+,20-/m1/s1
InChI key:InChIKey=STBZIDOIKQNFCQ-HSALFYBXSA-N
SMILES:O[C@@]12[C@@]3(C=4C(C[C@]1(N(CC5CC5)CC3)[H])=CC=C(O)C4)CCCC2
Synonyms:
  • Oxilorphanum
  • Oxilorphanum [INN-Latin]
  • Oxilorfano
  • UNII-9Y9J2J74TO
  • Oxilorphan [USAN:INN]
  • Oxilorphane [INN-French]
  • Oxilorphan
  • Morphinan-3,14-diol, 17-(cyclopropylmethyl)-
  • Oxilorphane
  • levo-BC 2605
  • See more synonyms
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  • Oxilorphan
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    Oxilorphan

    CAS:
    Oxilorphan is a μ-opioid blocker and a weak κ-opioid activator; similar to naloxone in strength; can cause hallucinations and dysphoria.
    Formula:C20H27NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:313.43

    Ref: TM-T25910