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CAS 4406-22-8

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Cyprenorphine

Description:
Cyprenorphine is a synthetic opioid that functions primarily as a potent analgesic and has been studied for its potential use in pain management. It is classified as a mixed agonist-antagonist, meaning it can activate certain opioid receptors while simultaneously blocking others, which may help reduce the risk of addiction and side effects commonly associated with full agonists. Cyprenorphine exhibits a high affinity for the mu-opioid receptor, contributing to its analgesic properties, while its antagonistic effects at the kappa-opioid receptor may mitigate dysphoria and other adverse effects. The compound is typically administered in a controlled setting due to its pharmacological effects and potential for abuse. In terms of physical properties, cyprenorphine is a white to off-white crystalline powder, and its solubility varies depending on the solvent used. As with many opioids, careful consideration of dosage and monitoring for side effects is essential in clinical applications. Overall, cyprenorphine represents a significant area of interest in opioid research, particularly in the context of developing safer pain management therapies.
Formula:C26H33NO4
InChI:InChI=1S/C26H33NO4/c1-23(2,29)18-13-24-8-9-26(18,30-3)22-25(24)10-11-27(14-15-4-5-15)19(24)12-16-6-7-17(28)21(31-22)20(16)25/h6-9,15,18-19,22,28-29H,4-5,10-14H2,1-3H3/t18-,19-,22-,24-,25+,26-/m1/s1
InChI key:InChIKey=VSKIOMHXEUHYSI-KNLIIKEYSA-N
SMILES:O(C)[C@@]12[C@]3([C@]45[C@@]([C@](N(CC6CC6)CC4)(CC7=C5C(O3)=C(O)C=C7)[H])(C[C@@H]1[C@@](C)(C)O)C=C2)[H]
Synonyms:
  • (5Beta,9Alpha,13Alpha)-17-(Cyclopropylmethyl)-18-(2-Hydroxypropan-2-Yl)-6-Methoxy-7,8-Didehydro-18,19-Dihydro-4,5-Epoxy-6,14-Ethenomorphinan-3-Ol
  • (5α,7α)-17-(Cyclopropylmethyl)-4,5-epoxy-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol
  • 2-(N-Cyclopropylmethyl-4,5-epoxy-6-methoxy-6,14-endo-morphinan-7alpha-yl)-2-propanol
  • 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-4,5-epoxy-3-hydroxy-6-methoxy-alpha,alpha-dimethyl-, (5alpha,7alpha)-
  • 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-4,5-epoxy-3-hydroxy-6-methoxy-α,α-dimethyl-, (5α,7α)-
  • 6,14-endo-Ethenotetrahydrooripavine, 21-cyclopropyl-7alpha-(1-hydroxy-1-methylethyl)-
  • 6,14-endo-Ethenotetrahydrooripavine, 21-cyclopropyl-7α-(1-hydroxy-1-methylethyl)-
  • Ciprenorfina
  • Ciprenorfina [INN-Spanish]
  • Cyprenorphine [INN:BAN]
  • See more synonyms
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Found 1 products.
  • Cyprenorphine
    TRC
    + Info

    Cyprenorphine

    Controlled Product
    CAS:
    Formula:C26H33NO4
    Color and Shape:Neat
    Molecular weight:423.545

    Ref: TR-C999645

    50mg
    8,684.00€