CAS 4682-36-4

Orphenadrine citrate

Description:

Orphenadrine citrate is a chemical compound primarily used as a muscle relaxant and an anticholinergic agent. It is classified as a diphenylmethane derivative and is known for its ability to alleviate muscle spasms and discomfort associated with musculoskeletal conditions. The substance acts by blocking certain neurotransmitters in the central nervous system, which helps reduce muscle stiffness and pain. Orphenadrine citrate is typically administered in its citrate salt form, enhancing its solubility and bioavailability. It is often used in combination with other medications to improve therapeutic outcomes. The compound is generally well-tolerated, but it may cause side effects such as dry mouth, dizziness, and sedation. Due to its anticholinergic properties, caution is advised in patients with conditions like glaucoma or urinary retention. As with any medication, it is essential to use orphenadrine citrate under medical supervision to ensure safety and efficacy.

Formula: C₂₄H₃₁NO₈

InChI: InChI=1S/C18H23NO.C6H8O7/c1-15-9-7-8-12-17(15)18(20-14-13-19(2)3)16-10-5-4-6-11-16;7-3(8)1-6(13,5(11)12)2-4(9)10/h4-12,18H,13-14H2,1-3H3;13H,1-2H2,(H,7,8)(H,9,10)(H,11,12)

InChI key: InChIKey=MMMNTDFSPSQXJP-UHFFFAOYSA-N

SMILES: C(OCCN(C)C)(C1=C(C)C=CC=C1)C2=CC=CC=C2.C(CC(O)=O)(CC(O)=O)(C(O)=O)O

Synonyms:

• Ethanamine, N,N-dimethyl-2-[(2-methylphenyl)phenylmethoxy]-, 2-hydroxy-1,2,3-propanetricarboxylate (1:1)
• Ethylamine, N,N-dimethyl-2-[(o-methyl-α-phenylbenzyl)oxy]-, citrate (1:1)
• Orphenadrine citrate
• Norflex (pharmaceutical)
• Plenactol
• orphenadrine dihydrogen citrate
• β-dimethylaminoethyl 2-methylbenzhydryl ether hydrochloride
• X-Otag
• Banflex
• BETA-DIMETHYLAMINOETHYL 2-METHYLBENZHYDRYL ETHER CITRATE SALT
• ORPHENADRINE CITRATE SALT
• Norflex
• ORPHENADRINECITRATE,USP
• o-methyldiphenhydramine citrate
• X-Ota
• beta-dimethylaminoethyl 2-methylbenzhydryl ether citrate

ORPHENADRINE CITRATE CRS

CAS: 4682-36-4

ORPHENADRINE CITRATE CRS

Formula: C₂₄H₃₁NO₈

Color and Shape: Crystalline Powder. White. Powder.

Molecular weight: 461.5048

Ref: 41-Y0000101

Orphenadrine Citrate

CAS: 4682-36-4

Aromatic drugs of amino-alcohols, other than those contg more than one kind of oxygen function, their ethers and esters; salts thereof, nesoi

Formula: C₁₈H₂₃NO·C₆H₈O₇

Color and Shape: White Crystalline Powder

Molecular weight: 269.17796

Ref: 45-1479009

Orphenadrine Citrate

CAS: 4682-36-4

Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.

Formula: C₁₈H₂₃NO·C₆H₈O₇

Purity: 98% - 99.58%

Color and Shape: White Solid

Molecular weight: 461.5

Ref: TM-T6618

Orphenadrine Citrate

CAS: 4682-36-4

Formula: C₁₈H₂₃NO·C₆H₈O₇

Color and Shape: White To Off-White Solid

Molecular weight: 269.39 192.12

Ref: 4Z-O-056

Orphenadrine Citrate

CAS: 4682-36-4

Orphenadrine Citrate

Purity: ≥98%

Molecular weight: 461.5g/mol

Ref: 54-BUP14782

Orphenadrine Citrate

Controlled Product

CAS: 4682-36-4

Formula: C₁₈H₂₃NO·C₆H₈O₇

Color and Shape: Neat

Molecular weight: 461.50

Ref: 86-MM3601.00

Obeticholic Acid Impurity 13

CAS: 4682-36-4

Formula: C₂₆H₄₂O₃

Molecular weight: 402.62

Ref: 4Z-O-056014

Orphenadrine Citrate

CAS: 4682-36-4

Formula: C₁₈H₂₃NOC₆H₈O₇

Molecular weight: 269.39 : 192.1

Ref: ST-EA-CP-O22011

Orphenadrine Citrate Salt

CAS: 4682-36-4

Applications Muscle relaxant (skeletal); antihistaminic.
References Harms, N., et al.: J. Med. Pharm. Chem., 2, 57 (1960),

Formula: C₁₈H₂₃NO·C₆H₈O₇

Color and Shape: Neat

Molecular weight: 461.50

Ref: TR-O695300

Orphenadrine-d3 Citrate Salt

Controlled Product

CAS: 1185011-75-9, 4682-36-4

Stability Hygroscopic and Moisture Sensitive
Applications Muscle relaxant (skeletal); antihistaminic.
References Harms, N., et al.: J. Med. Pharm. Chem., 2, 57 (1960)

Formula: C₂₄H₂₈D₃NO₈

Color and Shape: Neat

Molecular weight: 464.52

Ref: TR-O695302

Orphenadrine citrate salt

Controlled Product

CAS: 4682-36-4

Orphenadrine citrate salt is a nonsteroidal anti-inflammatory drug that is used to treat pain and inflammation. It is also used in the treatment of cancer, as well as in the prevention of side effects associated with chemotherapy. Orphenadrine citrate salt is primarily used to relieve muscle spasms and to reduce pain, especially in cases of cancer. This medication has been shown to be effective for treating cervical cancer, psychiatric patients, and geriatric patients. Orphenadrine citrate salt has also been found to have antibiotic properties against bacteria such as capsicum annuum and other drugs that are metabolized by the liver.

Formula: C₂₄H₃₁NO₈

Purity: Min. 95%

Color and Shape: White To Off-White Solid

Molecular weight: 461.5 g/mol

Ref: 3D-FO26587

Ethanamine, N,N-dimethyl-2-[(2-methylphenyl)phenylmethoxy]-,2-hydroxy-1,2,3-propanetricarboxylate (1:1)

CAS: 4682-36-4

Formula: C₂₄H₃₁NO₈

Color and Shape: Solid

Molecular weight: 461.5048

Ref: IN-DA019FSG