CAS 475115-35-6

Galnon

Description:

Galnon, with the CAS number 475115-35-6, is a chemical compound that belongs to the class of small molecules. It is primarily recognized for its role as a selective antagonist of certain receptors, particularly in the context of pharmacological research. The compound exhibits specific binding affinity, which makes it a valuable tool in studying receptor functions and potential therapeutic applications. Galnon's molecular structure includes functional groups that contribute to its biological activity, although detailed information about its physical properties, such as solubility, melting point, and stability, may vary based on the specific formulation and conditions. As with many chemical substances, safety data sheets and handling guidelines should be consulted to ensure proper usage and to understand any potential hazards associated with the compound. Overall, Galnon represents a significant interest in medicinal chemistry, particularly in the exploration of new treatments for various conditions.

Formula: C₄₀H₄₆N₄O₆

InChI: InChI=1S/C40H46N4O6/c1-25-21-37(45)50-36-23-27(18-19-28(25)36)42-38(46)34(17-9-10-20-41)43-39(47)35(22-26-11-3-2-4-12-26)44-40(48)49-24-33-31-15-7-5-13-29(31)30-14-6-8-16-32(30)33/h5-8,13-16,18-19,21,23,26,33-35H,2-4,9-12,17,20,22,24,41H2,1H3,(H,42,46)(H,43,47)(H,44,48)/t34-,35-/m0/s1

InChI key: InChIKey=IKNOZZKXIDSTRN-PXLJZGITSA-N

SMILES: C(OC(N[C@@H](CC1CCCCC1)C(N[C@H](C(NC=2C=C3C(=CC2)C(C)=CC(=O)O3)=O)CCCCN)=O)=O)C4C=5C(C=6C4=CC=CC6)=CC=CC5

Synonyms:

• 3-Cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-<span class="text-smallcaps">L</smallcap>-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-<smallcap>L</span>-lysinamide
• 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-chromen-7-yl)-L-lysinamide
• <span class="text-smallcaps">L</smallcap>-Lysinamide, 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-<smallcap>L</span>-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-
• Galnon
• L-Lysinamide, 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-
• 3-Cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-L-lysinamide

Galnon

CAS: 475115-35-6

The galanin receptor agonist galnon binds to the same brain-surface proteins, or receptors, that galanin does and prevents seizures. This drug mimicking a natural substance in the brain may represent a prototype for a new class of epilepsy drugs.

Formula: C₄₀H₄₆N₄O₆

Purity: 98.3%

Color and Shape: White Powder

Molecular weight: 678.83

Ref: 01-4040530

GALNON

CAS: 475115-35-6

Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties

Formula: C₄₀H₄₆N₄O₆

Purity: 98%

Color and Shape: Solid

Molecular weight: 678.82

Ref: TM-T8456

Galnon trifluoroacetate salt

CAS: 475115-35-6

Galnon trifluoroacetate salt is a pharmacological agent that binds to galanin and inhibits its binding to G protein-coupled receptors. It was shown to have a cancer preventive effect on 3T3-L1 preadipocytes by inhibiting the production of the inflammatory cytokine, tumor necrosis factor-α (TNF-α). Galnon trifluoroacetate salt also has an effect on the immune system and may be used as an anti-inflammatory agent in autoimmune diseases. This drug has been shown to block the effects of galanin on camp levels, leading to a decrease in locomotor activity.

Formula: C₄₀H₄₆N₄O₆

Purity: Min. 95%

Molecular weight: 678.82 g/mol

Ref: 3D-FG111343