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CAS 478296-72-9

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Gabapentin enacarbil

Description:
Gabapentin enacarbil is a prodrug of gabapentin, primarily used for the treatment of neuropathic pain and restless legs syndrome. It is characterized by its ability to enhance the bioavailability of gabapentin, allowing for improved absorption and therapeutic efficacy. The chemical structure of gabapentin enacarbil includes an enacarbil moiety that facilitates its conversion to gabapentin in the body. This compound is typically administered orally and is known for its relatively favorable safety profile, with common side effects including dizziness, fatigue, and somnolence. Gabapentin enacarbil acts by modulating the release of excitatory neurotransmitters, thereby reducing neuronal excitability. Its pharmacokinetics are influenced by factors such as food intake, which can affect absorption rates. Overall, gabapentin enacarbil represents a significant advancement in the management of certain neurological conditions, providing an alternative for patients who may not respond adequately to traditional gabapentin therapy.
Formula:C16H27NO6
InChI:InChI=1S/C16H27NO6/c1-11(2)14(20)22-12(3)23-15(21)17-10-16(9-13(18)19)7-5-4-6-8-16/h11-12H,4-10H2,1-3H3,(H,17,21)(H,18,19)
InChI key:InChIKey=TZDUHAJSIBHXDL-UHFFFAOYSA-N
SMILES:C(NC(OC(OC(C(C)C)=O)C)=O)C1(CC(O)=O)CCCCC1
Synonyms:
  • 1-[[(1-(Isobutanoyloxy)ethoxy)carbonyl]aminomethyl]cyclohex-1-ylacetic acid
  • Cyclohexaneacetic acid, 1-[[[[1-(2-methyl-1-oxopropoxy)ethoxy]carbonyl]amino]methyl]-
  • Gabapentin enacarbil
  • Horizant
  • Regnite
  • Xp 13512
  • 1-[[[[1-(2-Methyl-1-oxopropoxy)ethoxy]carbonyl]amino]methyl]cyclohexaneacetic acid
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