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CAS 486-16-8

:

(±)-Carbinoxamine

Description:
(±)-Carbinoxamine is an antihistamine with anticholinergic properties, primarily used to alleviate allergy symptoms. It is classified as a first-generation antihistamine, which means it can cross the blood-brain barrier, often leading to sedation as a side effect. The substance is a racemic mixture, containing both enantiomers, which can exhibit different pharmacological effects. Its chemical structure includes a piperidine ring, contributing to its activity as a histamine H1 receptor antagonist. (±)-Carbinoxamine is typically administered orally and is effective in treating allergic rhinitis, urticaria, and other allergic conditions. The compound is also known for its potential to cause side effects such as dry mouth, dizziness, and drowsiness, which are common among first-generation antihistamines. Due to its sedative effects, caution is advised when operating machinery or driving after consumption. Additionally, it is important to consider drug interactions, especially with other central nervous system depressants. Overall, (±)-Carbinoxamine serves as a useful therapeutic agent in managing allergic reactions, albeit with a profile that necessitates careful monitoring of its effects.
Formula:C16H19ClN2O
InChI:InChI=1/C16H19ClN2O/c1-19(2)11-12-20-16(15-5-3-4-10-18-15)13-6-8-14(17)9-7-13/h3-10,16H,11-12H2,1-2H3
InChI key:InChIKey=OJFSXZCBGQGRNV-UHFFFAOYSA-N
SMILES:C(OCCN(C)C)(C1=CC=C(Cl)C=C1)C2=CC=CC=N2
Synonyms:
  • 2-(4-Chloro-Alpha-(2-Pyridyl)Benzyloxy)Ethyldimethylamine
  • 2-[(4-Chlorophenyl)-2-Pyridinylmethoxy]-N,N-Dimethylethanamine
  • 2-[P-Chloro-A-(2-Dimethylaminoethoxy)Benzyl]Pyridine
  • 2-[p-Chloro-α-[2-(dimethylamino)ethoxy]benzyl]pyridine
  • Carbinoxamin
  • Carbinoxamina
  • Carbinoxamine (base and/or unspecified salts)
  • Ethanamine, 2-[(4-chlorophenyl)-2-pyridinylmethoxy]-N,N-dimethyl-
  • McN-R 73Z
  • Paracarbinoxamine
  • See more synonyms
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