CAS 51931-66-9
:Tilidine
Description:
Tilidine is a synthetic opioid analgesic primarily used for the management of moderate to severe pain. It is classified as a prodrug, meaning it is metabolized in the body to its active form, nortilidine, which exerts the analgesic effects. Tilidine acts on the central nervous system by binding to opioid receptors, leading to pain relief. Its chemical structure includes a phenylpiperidine moiety, which is characteristic of many opioids. The substance is typically administered in combination with naloxone to mitigate the risk of misuse and to prevent potential opioid-related side effects. Tilidine has a relatively rapid onset of action and a moderate duration of effect, making it suitable for various pain management scenarios. However, like other opioids, it carries risks of dependence, tolerance, and withdrawal symptoms. Due to its potential for abuse, tilidine is regulated in many countries, and its use is often restricted to specific medical contexts.
Formula:C17H23NO2
InChI:InChI=1/C17H23NO2/c1-4-20-16(19)17(14-10-6-5-7-11-14)13-9-8-12-15(17)18(2)3/h5-8,10-12,15H,4,9,13H2,1-3H3/t15-,17+/m1/s1
InChI key:InChIKey=WDEFBBTXULIOBB-XELGSYHNNA-N
SMILES:C(OCC)(=O)[C@]1([C@H](N(C)C)C=CCC1)C2=CC=CC=C2
Synonyms:- 3-Cyclohexene-1-carboxylic acid, 2-(dimethylamino)-1-phenyl-, ethyl ester, (1R,2S)-rel-
- 3-Cyclohexene-1-carboxylic acid, 2-(dimethylamino)-1-phenyl-, ethyl ester, trans-
- Ethyl trans-2-(dimethylamino)-1-phenyl-3-cyclohexene-1-carboxylate
- Tilidate [BAN]
- Tilidine
- Tilidine [USAN:INN]
- dl-trans-Tilidine
- trans-Tilidine
- Ethyl trans-2-(dimethylamino)-1-phenylcyclohex-3-ene-1-carboxylate
- Einecs 257-522-9
- Dea no. 9750
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