CAS 53251-94-8

Pinaverium bromide

Description:

Pinaverium bromide is a synthetic compound primarily used as an antispasmodic agent, particularly in the treatment of gastrointestinal disorders. It functions by inhibiting the activity of calcium channels, which helps to relax smooth muscle and alleviate spasms in the digestive tract. The substance is characterized by its bromide salt form, which enhances its solubility and bioavailability. Pinaverium bromide is typically administered orally and is known for its relatively low side effect profile compared to other antispasmodics. Its chemical structure includes a quaternary ammonium group, contributing to its pharmacological properties. The compound is generally well-tolerated, but like any medication, it may cause adverse effects in some individuals, such as dry mouth or constipation. It is important for patients to consult healthcare professionals before use, especially if they have underlying health conditions or are taking other medications. Overall, pinaverium bromide is a valuable therapeutic option for managing gastrointestinal motility disorders.

Formula: C₂₆H₄₁Br₂NO₄

InChI: InChI=1/C26H41BrNO4.BrH/c1-26(2)21-6-5-19(22(26)16-21)7-11-31-12-8-28(9-13-32-14-10-28)18-20-15-24(29-3)25(30-4)17-23(20)27;/h15,17,19,21-22H,5-14,16,18H2,1-4H3;1H/q+1;/p-1

InChI key: InChIKey=IKGXLCMLVINENI-UHFFFAOYSA-M

SMILES: C([N+]1(CCOCCC2C3C(C)(C)C(C3)CC2)CCOCC1)C4=CC(OC)=C(OC)C=C4Br.[Br-]

Synonyms:

• 258-450-0
• 4-(2-Bromo-4,5-Dimethoxybenzyl)-4-{2-[2-(6,6-Dimethylbicyclo[3.1.1]Hept-2-Yl)Ethoxy]Ethyl}Morpholin-4-Ium Bromide
• 4-(6-Bromoveratryl)-4-[2-[2-(6,6-dimethyl-2-norpinyl)ethoxy]ethyl]morpholinium Bromide
• 4-[(2-Bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]morpholinium Bromide
• 53251-94-8
• <span class="text-smallcaps">L</span>-Pinaverium bromide
• Dicetel
• Eldicet
• Lat 1717
• Morpholinium, 4-[(2-bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-, bromide
• Morpholinium, 4-[(2-bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-, bromide (1:1)
• Pinaverium bromide
• 4-[(2-Bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(7,7-dimethyl-2-bicyclo[3.1.1]heptanyl)ethoxy]ethyl]morpholin-4-ium bromide
• 4-(2-Bromo-4,5-dimethoxybenzyl-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]heptan-2-yl)ethoxy]ethyl]morpholinium bromide
• L-Pinaverium bromide
• PINAVERIUM BROMIDE-D4
• morpholin-4-ium bromide
• 4-(2-Bromo-4,5-dimethoxybenzyl)-4-(2-(2-(6,6-dimethylbicyclo[3.1.1]heptan-2-yl)ethoxy)ethyl)morpholin-4-ium bromide
• Pinaverium
• 4-(2-Bromo-4,5-dimethoxybenzyl)
• 4-[(2-Bromo-4,5-dimethoxy-phenyl)methyl]-4-[2-[2-(6,6-dimethylnorpinan-2-yl)ethoxy]ethyl]-1-oxa-4-azoniacyclohexane bromide
• Pinaverium bromide (inn)
• -4-(2-(2-(6,6-dimethylbicyclo[3.1.1]heptan-2-yl)
• Morpholinium, 4-[(2-bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-
• 4-[(2-Bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-, bromide

Pinaverium Bromide

CAS: 53251-94-8

Formula: C₂₆H₄₁BrNO₄Br

Molecular weight: 511.5 : 79.9

Ref: ST-EA-CP-P35005

Morpholinium,4-[(2-bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-, bromide

CAS: 53251-94-8

Formula: C₂₆H₄₁Br₂NO₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 591.4160

Ref: IN-DA00I9I8

4-[(2-Bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-Morpholinium bromide (1:1)

CAS: 53251-94-8

4-[(2-Bromo-4,5-dimethoxyphenyl)methyl]-4-[2-[2-(6,6-dimethylbicyclo[3.1.1]hept-2-yl)ethoxy]ethyl]-Morpholinium bromide (1:1)

Purity: 99%

Molecular weight: 591.42g/mol

Ref: 54-OR317274

Pinaverium-d4 Bromide (Mixture of Diastereomers)

CAS: 53251-94-8

Formula: C₂₆H₃₇D₄BrNO₄·Br

Color and Shape: White To Off-White Solid

Molecular weight: 515.55 79.90

Ref: 4Z-P-706

Pinaverium Bromide (Mixture of Diastereomers)

CAS: 53251-94-8

Formula: C₂₆H₄₁BrNO₄·Br

Color and Shape: White To Off-White Solid

Molecular weight: 511.52 79.90

Ref: 4Z-P-701

Pinaverium bromide

CAS: 53251-94-8

Pinaverium bromide

Purity: ≥98%

Molecular weight: 591.42g/mol

Ref: 54-BUP15656

Pinaverium Bromide

CAS: 53251-94-8

Formula: C₂₆H₄₁Br₂NO₄

Purity: >98.0%(T)(HPLC)

Color and Shape: White to Light yellow powder to crystal

Molecular weight: 591.43

Ref: 3B-P2753

Pinaverium bromide

CAS: 53251-94-8

Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.

Formula: C₂₆H₄₁Br₂NO₄

Purity: 99.52%

Color and Shape: White Crystalline Powder

Molecular weight: 591.42

Ref: TM-T7603

Pinaverium Bromide

CAS: 53251-94-8

Applications Spasmolytic agent with low incidence of anticholinergic effects. Antispasmodic.
References Jacquot, C., et al.: Eur. J. Med. Chem., 13, 61 (1978), Bretaudeau, J., et al.: J. Pharmacol., 11, 233 (1980), Bertrand, J., et al.: Therapie, 36, 555 (1981),

Formula: C₂₆H₄₁BrNO₄·Br

Color and Shape: Neat

Molecular weight: 591.42

Ref: TR-P465000

Pinaverium Bromide

CAS: 53251-94-8

Purity: 98%

Molecular weight: 591.4249878

Ref: 10-F876149

Pinaverium-d4 Bromide

Controlled Product

CAS: 53251-94-8

Applications Spasmolytic agent with low incidence of anticholinergic effects. Antispasmodic.
References Jacquot, C., et al.: Eur. J. Med. Chem., 13, 61 (1978), Bretaudeau, J., et al.: J. Pharmacol., 11, 233 (1980), Bertrand, J., et al.: Therapie, 36, 555 (1981),

Formula: C₂₆D₄H₃₇BrNO₄·Br

Color and Shape: Neat

Molecular weight: 595.441

Ref: TR-P465002

Pinaverium bromide

CAS: 53251-94-8

Pinaverium bromide is a drug with anti-inflammatory properties. It is used in the treatment of bowel disease and as a muscle relaxant. Pinaverium bromide has shown efficacy in treating bowel syndrome, but it also reduces blood flow to the bowel. Pinaverium bromide inhibits voltage-dependent calcium channels, leading to muscle relaxation. This drug also has been shown to inhibit the production of inflammatory mediators such as prostaglandins and leukotrienes, which may be due to its ability to inhibit basic fibroblast growth factor production. Pinaverium bromide is an effective drug that is used for the treatment of bowel disease and muscle spasms. It blocks voltage-dependent calcium channels, which leads to muscle relaxation without affecting heart function. The inhibition of basic fibroblast growth factor production may contribute to this drug's anti-inflammatory effects.!-- START: Description --> Pinaverium bromide

Formula: C₂₆H₄₁Br₂NO₄

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 591.42 g/mol

Ref: 3D-FP27052