CAS 54340-62-4

Bufuralol

Description:

Bufuralol is a pharmaceutical compound primarily recognized for its role as a non-selective beta-adrenergic antagonist, which means it can block the action of certain neurotransmitters on beta receptors in the body. This compound is often utilized in the treatment of hypertension and certain cardiac conditions due to its ability to reduce heart rate and lower blood pressure. Bufuralol exhibits a unique characteristic of having both beta-blocking and mild vasodilatory effects, which can enhance its therapeutic efficacy. The substance is classified as a secondary amine and has a specific stereochemistry that contributes to its pharmacological properties. Its solubility profile indicates that it is moderately soluble in water, which is relevant for its formulation in pharmaceutical preparations. Additionally, bufuralol's metabolism involves hepatic pathways, and it is known to have a variable half-life depending on individual patient factors. Overall, bufuralol's multifaceted action makes it a valuable agent in cardiovascular therapy, although its use must be carefully monitored due to potential side effects associated with beta-blockers.

Formula: C₁₆H₂₃NO₂

InChI: InChI=1S/C16H23NO2/c1-5-11-7-6-8-12-9-14(19-15(11)12)13(18)10-17-16(2,3)4/h6-9,13,17-18H,5,10H2,1-4H3

InChI key: InChIKey=SSEBTPPFLLCUMN-UHFFFAOYSA-N

SMILES: C(C)C1=C2C(C=C(C(CNC(C)(C)C)O)O2)=CC=C1

Synonyms:

• dl-Bufuralol
• Ro 3-4787
• Bufuralol
• 2-Benzofuranmethanol, α-[[(1,1-dimethylethyl)amino]methyl]-7-ethyl-
• α-[[(1,1-Dimethylethyl)amino]methyl]-7-ethyl-2-benzofuranmethanol

Bufuralol

CAS: 54340-62-4

Formula: C₁₆H₂₃NO₂

Molecular weight: 261.37

Ref: 4Z-B-251

Bufuralol

CAS: 54340-62-4

Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.

Formula: C₁₆H₂₃NO₂

Purity: 98.26%

Color and Shape: Solid

Molecular weight: 261.36

Ref: TM-T30611