CAS 55974-42-0

1,3(2H,4H)-Isoquinolinedione,2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-4,4-dimethyl-,dihydrochloride

Description:

1,3(2H,4H)-Isoquinolinedione, 2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-4,4-dimethyl-, dihydrochloride, with CAS number 55974-42-0, is a chemical compound characterized by its complex structure, which includes an isoquinoline core and a piperazine moiety. This compound typically exhibits properties associated with its functional groups, such as potential pharmacological activity, making it of interest in medicinal chemistry. The presence of the methoxyphenyl group may enhance lipophilicity, influencing its bioavailability and interaction with biological targets. As a dihydrochloride salt, it is likely to be more soluble in water compared to its free base form, which is advantageous for formulation in pharmaceutical applications. The compound may also exhibit specific reactivity patterns due to the presence of the isoquinoline and piperazine rings, which can participate in various chemical reactions. Overall, this compound's unique structural features suggest potential utility in drug development, particularly in the context of neuropharmacology or other therapeutic areas.

Formula: C₂₄H₃₀ClN₃O₃

Synonyms:

• Adrenergic Receptor,adrenoceptor antagonist,inhibit,ARC 239,Beta Receptor,ARC239,BHT-920,ARC 239 dihydrochloride,UK 14,304,ARC-239,pig nasal mucosa,Inhibitor,phenylephrine

ARC 239 dihydrochloride

CAS: 55974-42-0

ARC 239 dihydrochloride

Purity: ≥98%

Molecular weight: 480.43g/mol

Ref: 54-BUP11537

ARC 239 dihydrochloride

CAS: 55974-42-0

ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).

Formula: C₂₄H₃₁Cl₂N₃O₃

Purity: 99.72%

Color and Shape: Solid

Molecular weight: 480.43

Ref: TM-T22033

ARC 239 Dihydrochloride

Controlled Product

CAS: 55974-42-0

Formula: C₂₄H₂₉N₃O₃•2(HCl)

Color and Shape: Neat

Molecular weight: 407.5123646

Ref: TR-A766573

ARC 239 Dihydrochloride

CAS: 55974-42-0

ARC 239 Dihydrochloride is a cholinergic drug that is used in the treatment of neurologic disorders. It has been shown to be effective in vivo in animal models of Parkinson's disease and dystonia, as well as clinical studies. ARC 239 Dihydrochloride binds to the GABAA receptor on postsynaptic neurons, inhibiting the influx of chloride ions and causing hyperpolarization. This drug also has been shown to inhibit the production of nitric oxide by suppressing NOS activity.

Formula: C₂₄H₂₉N₃O₃·2HCl

Purity: Min. 95%

Molecular weight: 480.43 g/mol

Ref: 3D-FCA97442