CAS 568580-02-9

YM-254890

CAS: 568580-02-9

YM-254890 blocks P2Y1, prevents ADP-induced platelet aggregation, and selectively inhibits Gαq/11 with IC50 < 0.6 μM. Not affecting other G proteins.

Formula: C₄₆H₆₉N₇O₁₅

Purity: 95%

Color and Shape: Solid

Molecular weight: 960.08

Ref: TM-T17273

YM-254890

CAS: 568580-02-9

YM-254890 is a potent inhibitor of protein α and alkoxy radical in the thrombin receptor. It has been shown to be effective in inhibiting blood pressure and α subunit, which is one of the main proteins involved in the regulation of blood pressure. YM-254890 is a hydrogenated analog that belongs to the class of non-selective cations. It also inhibits protein synthesis, which may be due to its binding to the carbonyl group and protein inhibitors. The biological properties of YM-254890 have been studied with carboxylic acid groups, including thrombin receptors, and it has been found that this drug can inhibit cancer cell growth.

Formula: C₄₆H₆₉N₇O₁₅

Purity: Min. 95%

Molecular weight: 960.1 g/mol

Ref: 3D-TXA58002