CAS 58662-84-3

Meclonazepam

Description:

Meclonazepam is a chemical compound belonging to the benzodiazepine class, characterized by its psychoactive properties. It is primarily known for its anxiolytic, sedative, and muscle relaxant effects. The molecular structure of Meclonazepam features a benzodiazepine core, which is essential for its biological activity, and it typically includes a chlorine atom and a methyl group that contribute to its pharmacological profile. This compound is often used in research settings to study its effects on the central nervous system, although it is not widely prescribed in clinical practice. Meclonazepam acts by enhancing the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased inhibitory neurotransmission. Due to its potential for dependence and abuse, it is classified as a controlled substance in many jurisdictions. Safety and toxicity profiles are important considerations, as with all benzodiazepines, and users should be aware of the risks associated with its use.

Formula: C₁₆H₁₂ClN₃O₃

InChI: InChI=1S/C16H12ClN3O3/c1-9-16(21)19-14-7-6-10(20(22)23)8-12(14)15(18-9)11-4-2-3-5-13(11)17/h2-9H,1H3,(H,19,21)/t9-/m0/s1

InChI key: InChIKey=LMUVYJCAFWGNSY-VIFPVBQESA-N

SMILES: ClC1=C(C=2C=3C(=CC=C(N(=O)=O)C3)NC(=O)[C@H](C)N2)C=CC=C1

Synonyms:

• (3S)-5-(2-Chlorophenyl)-1,3-dihydro-3-methyl-7-nitro-2H-1,4-benzodiazepin-2-one
• (3S)-5-(2-Chlorophenyl)-3-methyl-7-nitro-1,3-dihydro-1,4-benzodiazepin-2-one
• (3S)-5-(2-Chlorophenyl)-3-methyl-7-nitro-1,3-dihydro-2H-1,4-benzodiazepin-2-one
• 2H-1,4-Benzodiazepin-2-one, 5-(2-chlorophenyl)-1,3-dihydro-3-methyl-7-nitro-, (S)-
• 2H-1,4-benzodiazepin-2-one, 5-(2-chlorophenyl)-1,3-dihydro-3-methyl-7-nitro-, (3S)-
• Ro 11-3128
• Ro 11-3128/002
• Meclonazepam

Meclonazepam-d4

Controlled Product

CAS: 58662-84-3

Formula: C₁₆D₄H₈ClN₃O₃

Color and Shape: Neat

Molecular weight: 333.762

Ref: TR-M202792

Meclonazepam

Controlled Product

CAS: 58662-84-3

Applications Meclonazepam, is a drug of a benzodiazepine class similar in structure to Clonazepam (C587080). It has sedative and anxiolytic properties. It has also shown to have anti-parasitic effects against the parasitic worm Schistosoma mansoni.
References O Boyle C., et al.: Euro. J. Clinic. Pharmacol., 29 (1), 105 (1985); Ansseau, M., et al.: Psychopharmacology, 87 (2), 130 (1985);

Formula: C₁₆H₁₂ClN₃O₃

Color and Shape: Off White Solid

Molecular weight: 329.74

Ref: TR-M202790

Meclonazepam

Controlled Product

CAS: 58662-84-3

Meclonazepam is a potent kinase inhibitor that has shown promising anticancer activity. It works by inducing apoptosis in cancer cells, leading to their death. Meclonazepam is an analog of the Chinese medicinal herb, and it has been found in human urine samples. This drug selectively inhibits kinases involved in tumor growth and progression, making it a potential therapeutic option for cancer treatment. Meclonazepam has been extensively studied for its inhibitory effects on various protein kinases and has shown significant promise as an effective anticancer agent. Its ability to induce apoptosis in cancer cells makes it a valuable tool in the fight against this deadly disease.

Formula: C₁₆H₁₂ClN₃O₃

Purity: Min. 95%

Molecular weight: 329.74 g/mol

Ref: 3D-ICA66284