CAS 58754-46-4

Iferanserin

Description:

Iferanserin, with the CAS number 58754-46-4, is a chemical compound that belongs to the class of serotonin receptor antagonists. It is primarily known for its potential applications in the treatment of various psychiatric and neurological disorders. The compound exhibits selective binding to specific serotonin receptors, which can influence neurotransmitter activity in the brain. Iferanserin is characterized by its unique molecular structure, which contributes to its pharmacological properties. It is typically administered in a controlled dosage form to ensure efficacy while minimizing side effects. The compound's solubility, stability, and reactivity are important factors that influence its formulation and therapeutic use. As with many pharmacologically active substances, understanding its mechanism of action, pharmacokinetics, and potential interactions with other drugs is crucial for its safe and effective application in clinical settings. Research continues to explore its full therapeutic potential and any associated risks.

Formula: C₂₃H₂₈N₂O

InChI: InChI=1S/C23H28N2O/c1-25-18-8-7-12-21(25)16-15-20-11-5-6-13-22(20)24-23(26)17-14-19-9-3-2-4-10-19/h2-6,9-11,13-14,17,21H,7-8,12,15-16,18H2,1H3,(H,24,26)/t21-/m0/s1

InChI key: InChIKey=UXIPFQUBOVWAQW-NRFANRHFSA-N

SMILES: C(C[C@H]1N(C)CCCC1)C2=C(NC(C=CC3=CC=CC=C3)=O)C=CC=C2

Synonyms:

• 2-Propenamide, N-[2-[2-(1-methyl-2-piperidinyl)ethyl]phenyl]-3-phenyl-, (-)-
• N-[2-[2-[(2S)-1-Methyl-2-piperidinyl]ethyl]phenyl]-3-phenyl-2-propenamide
• 2-Propenamide, N-[2-[2-[(2S)-1-methyl-2-piperidinyl]ethyl]phenyl]-3-phenyl-
• Iferanserin

Iferanserin

CAS: 58754-46-4

Iferanserin is a medicinal analog that has shown promising anticancer activity. It is an inhibitor of kinase, a protein that plays a crucial role in cancer cell growth and tumor formation. Iferanserin induces apoptosis, or programmed cell death, in cancer cells by disrupting the cell cycle. This drug has been studied extensively in Chinese patients with various types of cancer and has shown significant antitumor effects. Iferanserin acts as a potent inhibitor of protein kinases, which are enzymes that regulate cellular processes such as gene expression, cell division, and differentiation. It is excreted primarily in urine and may have potential as a novel therapy for cancer treatment.

Formula: C₂₃H₂₈N₂O

Purity: Min. 95%

Molecular weight: 348.5 g/mol

Ref: 3D-ICA75446

Iferanserin

CAS: 58754-46-4

Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.

Formula: C₂₃H₂₈N₂O

Color and Shape: Solid

Molecular weight: 348.48

Ref: TM-T15552