CAS 58786-99-5: Butorphanol tartrate
Description:Butorphanol tartrate is a synthetic opioid analgesic primarily used for pain management. It is classified as a mixed agonist-antagonist, meaning it can activate certain opioid receptors while simultaneously blocking others, which can help reduce the risk of dependence and respiratory depression associated with traditional opioids. The substance is typically administered via injection or nasal spray and is known for its relatively rapid onset of action. Butorphanol tartrate exhibits a higher affinity for the kappa-opioid receptor compared to the mu-opioid receptor, contributing to its analgesic effects. It is also characterized by its solubility in water, which facilitates its formulation for medical use. Common side effects may include sedation, dizziness, and nausea, and it is important to monitor patients for potential adverse reactions. Due to its opioid nature, butorphanol tartrate is classified as a controlled substance in many jurisdictions, necessitating careful prescribing and dispensing practices.
Formula:C21H29NO2·C4H6O6
InChI:InChI=1S/C21H29NO2.C4H6O6/c23-17-7-6-16-12-19-21(24)9-2-1-8-20(21,18(16)13-17)10-11-22(19)14-15-4-3-5-15;5-1(3(7)8)2(6)4(9)10/h6-7,13,15,19,23-24H,1-5,8-12,14H2;1-2,5-6H,(H,7,8)(H,9,10)/t19-,20+,21-;1-,2-/m10/s1
InChI key:InChIKey=GMTYREVWZXJPLF-AFHUBHILSA-N
SMILES:O=C(O)C(O)C(O)C(=O)O.OC1=CC=C2C(=C1)C34CCN(CC5CCC5)C(C2)C4(O)CCCC3
- Synonyms:
- 17-(Cyclobutylmethyl)Morphinan-3,14-Diol 2,3-Dihydroxybutanedioate (Salt)
- 17-(Cyclobutylmethyl)Morphinan-3,14-Diol 2,3-Dihydroxybutanedioate (1:1)
- [S-(R*,R*)]-2,3-dihidroxisuccinato de 17-(ciclobutilmetil)morfinan-3,14-diilo
- [S-(R*,R*)]-2,3-dihydroxysuccinate de 17-(cyclobutylmethyl)morphinan-3,14-diyle
- 17-(cyclobutylmethyl)morphinan-3,14-diyl [S-(R*,R*)]-2,3-dihydroxysuccinate
- 17-(Cyclobutylmethyl)morphinan-3,14-diyl-[S-(R*,R*)]-2,3-dihydroxysuccinat
- Butorphanol tartrate
- Butorphic
- l-Butorphanol tartrate
- Levo-BC 2627 tartrate
- See more synonyms
- Moradol
- Morphinan-3,14-diol, 17-(cyclobutylmethyl)-, (2S,3S)-2,3-dihydroxybutanedioate (1:1)
- Morphinan-3,14-diol, 17-(cyclobutylmethyl)-, (2S,3S)-2,3-dihydroxybutanedioate (1:1) (salt)
- Morphinan-3,14-diol, 17-(cyclobutylmethyl)-, [S-(R*,R*)]-2,3-dihydroxybutanedioate (1:1) (salt)
- Nih 10275
- Stadol
- Torate
- Torbugesic
Brand | Product data | Purity | Price range | Estimated delivery |
---|---|---|---|---|
![]() | Butorphanol Tartrate REF: 86-MM1192.00CAS: 58786-99-5 | - - - | 1,813.00 € | Thu 17 Apr 25 |
![]() | Butorphanol tartrate REF: 3D-ICA78699CAS: 58786-99-5 | Min. 95% | 188.00 €~1,005.00 € | Fri 25 Apr 25 |
![]() | Butorphanol Tartrate CIV REF: 45-1082504CAS: 58786-99-5 | - - - | To inquire | Tue 10 Jun 25 |

Butorphanol Tartrate
Controlled ProductRef: 86-MM1192.00
100mg | 1,813.00 € |

Butorphanol tartrate
Controlled ProductRef: 3D-ICA78699
10mg | 264.00 € | ||
25mg | 465.00 € | ||
50mg | 663.00 € | ||
100mg | 1,005.00 € |

Butorphanol Tartrate CIV
Controlled ProductRef: 45-1082504
350mg | To inquire |