CAS 5985-35-3

17-methylmorphinan-3-ol

Description:

17-Methylmorphinan-3-ol, also known as morphinan-3-ol, is an organic compound that belongs to the class of morphinans, which are bicyclic compounds derived from morphine. This substance is characterized by its structural features, including a hydroxyl group (-OH) at the 3-position and a methyl group at the 17-position of the morphinan skeleton. It exhibits analgesic properties and is often studied for its potential use in pain management and as a cough suppressant. The compound has a complex interaction with opioid receptors, primarily acting as a partial agonist. Its solubility profile typically indicates moderate solubility in organic solvents and limited solubility in water, which can influence its pharmacokinetics and bioavailability. Additionally, 17-methylmorphinan-3-ol may undergo metabolic transformations in the body, leading to various metabolites that can also exhibit biological activity. As with many morphinan derivatives, safety and regulatory considerations are important, particularly regarding its potential for abuse and dependence.

Formula: C₁₇H₂₃NO

InChI: InChI=1/C17H23NO/c1-18-9-8-17-7-3-2-4-14(17)16(18)10-12-5-6-13(19)11-15(12)17/h5-6,11,14,16,19H,2-4,7-10H2,1H3

SMILES: CN1CCC23CCCCC2C1Cc1ccc(cc31)O

Synonyms:

• 2H-10,4a-(Iminoethano)phenanthren-6-ol, 1,3,4,9,10,10a-hexahydro-11-methyl-, (+)-

Racemorphan Hydrobromide

Controlled Product

CAS: 5985-35-3

Stability Hygroscopic
Applications (±)-17-Methyl-morphinan-3-ol Hydrobromide is a racemic mixture of Dextrorphan Tartrate Salt (D299485) and Levorphanol Tartrate (L376500). Dextrorphan Tartrate Salt and Levorphanol Tartrate are orally active synthetic morphine analogs and analgesics (narcotic). Levorphanol Tartrate is a controlled substance.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Tallarida, R., et al.: Life Sci., 45, 947 (1989); Netzer, R., et al.: Eur. J. Pharmacol., 238, 209 (1993); Mao, J., et al.: Pain, 67, 361 (1996); Chow, L., et al.: J. Biomed. Sci., 11, 717 (2004); Randall, L.O., et al.: J. Pharmacol. Exp. Ther., 99, 163 (1950); Dajani, E., et al.: Eur. J. Pharmacol., 34, 105 (1975); Winpenny, J., et al.: Drugs, 8, 416 (2005),

Formula: C₁₇H₂₄BrNO

Color and Shape: Neat

Molecular weight: 338.28

Ref: TR-M321495

Racemorphan Hydrobromide (1 mg/mL in Methanol)

Controlled Product

CAS: 5985-35-3

Formula: C₁₇H₂₄BrNO

Color and Shape: Single Solution

Molecular weight: 338.28

Ref: TR-KIT8615