CAS 609799-22-6: Tasimelteon

Description: Tasimelteon is a synthetic compound primarily recognized for its role as a melatonin receptor agonist, specifically targeting the MT1 and MT2 receptors. It is classified as a non-benzodiazepine sleep aid and is primarily used in the treatment of circadian rhythm sleep disorders, particularly in individuals who are blind and experience non-24-hour sleep-wake disorder. The molecular formula of Tasimelteon reflects its complex structure, which includes multiple functional groups that contribute to its pharmacological activity. The substance is typically administered orally and has a relatively short half-life, necessitating careful dosing to achieve desired therapeutic effects. Its efficacy is attributed to its ability to mimic the action of melatonin, a hormone that regulates sleep-wake cycles. Additionally, Tasimelteon has undergone various clinical trials to assess its safety and effectiveness, demonstrating a favorable profile for managing sleep-related issues without the sedative side effects commonly associated with traditional sleep medications. As with any pharmacological agent, potential side effects and contraindications should be considered when prescribing Tasimelteon.

Formula: C₁₅H₁₉NO₂

InChI: InChI=1S/C15H19NO2/c1-2-15(17)16-9-10-8-13(10)11-4-3-5-14-12(11)6-7-18-14/h3-5,10,13H,2,6-9H2,1H3,(H,16,17)/t10-,13+/m0/s1

InChI key: InChIKey=PTOIAAWZLUQTIO-GXFFZTMASA-N

SMILES: O=C(NCC1CC1C=2C=CC=C3OCCC32)CC

Synonyms:

• (1R-trans)-N-[[2-(2,3-Dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide
• Bms 214778
• Hetlioz
• N-[[(1R,2R)-2-(2,3-Dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide
• N-{[(1R,2R)-2-(2,3-dihydro-1-benzofuran-4-yl)cyclopropyl]methyl}propanamide
• Propanamide, N-[[(1R,2R)-2-(2,3-dihydro-4-benzofuranyl)cyclopropyl]methyl]-
• Vec 162
• MA 1

Tasimelteon

CAS: 609799-22-6

• Formula: C₁₅H₁₉NO₂
• Purity: 97%
• Color and Shape: Solid
• Molecular weight: 245.3169

Tasimelteon

CAS: 609799-22-6

• Formula: C₁₅H₁₉NO₂
• Color and Shape: Off-White Solid
• Molecular weight: 245.32

Tasimelteon

CAS: 609799-22-6

• Formula: C₁₅H₁₉NO₂
• Purity: >95.0%(qNMR)
• Color and Shape: White to Almost white powder to crystal
• Molecular weight: 245.32

Tasimelteon

CAS: 609799-22-6

Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 …

• Formula: C₁₅H₁₉NO₂
• Purity: 98.08% - 99.93%
• Color and Shape: Solid
• Molecular weight: 245.32

Tasimelteon

CAS: 609799-22-6

Applications Tasimelteon is a novel drug, used in the treatment of non-24 hour sleep-wake disorder. …

• Formula: C₁₅H₁₉NO₂
• Color and Shape: Neat
• Molecular weight: 245.3169

Tasimelteon

CAS: 609799-22-6

Tasimelteon is a melatonin agonist that is used to treat insomnia in the elderly. It …

• Formula: C₁₅H₁₉NO₂
• Purity: Min. 95%
• Molecular weight: 245.32 g/mol