CAS 6440-42-2

2H-Benzimidazol-2-one, 1-[1-[1-(4-fluorophenyl)ethyl]-4-piperidinyl]-1,3-dihydro-

Description:

2H-Benzimidazol-2-one, 1-[1-[1-(4-fluorophenyl)ethyl]-4-piperidinyl]-1,3-dihydro- is a chemical compound characterized by its complex structure, which includes a benzimidazole core and a piperidine moiety. This compound typically exhibits properties associated with both the benzimidazole and piperidine functional groups, such as potential biological activity and solubility in organic solvents. The presence of a fluorophenyl group suggests that it may have enhanced lipophilicity and could interact with biological targets, making it of interest in medicinal chemistry. The compound may also exhibit specific pharmacological properties, potentially acting as a ligand for various receptors or enzymes. Its molecular structure allows for various stereochemical configurations, which can influence its biological activity and pharmacokinetics. As with many compounds in this class, it is essential to consider its safety profile, including toxicity and environmental impact, during research and application. Overall, this compound represents a class of substances that may have significant implications in drug development and therapeutic applications.

Formula: C₂₀H₂₂FN₃O

Synonyms:

• 2H-Benzimidazol-2-one, 1-[1-[1-(4-fluorophenyl)ethyl]-4-piperidinyl]-1,3-dihydro-

Fluorphine

CAS: 6440-42-2

Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.

Formula: C₂₀H₂₂FN₃O

Color and Shape: Solid

Molecular weight: 339.41

Ref: TM-T203493