CymitQuimica logo

CAS 65807-03-6

:

(D-Ser6)-Goserelin

Description:
(D-Ser6)-Goserelin is a synthetic peptide and a potent agonist of gonadotropin-releasing hormone (GnRH). It is primarily used in the treatment of hormone-sensitive conditions such as prostate cancer and endometriosis. The structure of (D-Ser6)-Goserelin includes a modified amino acid, D-Serine, which enhances its stability and bioactivity compared to natural GnRH. This modification allows for a prolonged half-life in the body, facilitating sustained suppression of gonadotropin release from the pituitary gland. The peptide acts by binding to GnRH receptors, leading to an initial surge in luteinizing hormone (LH) and follicle-stimulating hormone (FSH) levels, followed by downregulation of these hormones with continuous administration. This results in decreased levels of sex hormones such as testosterone and estrogen. (D-Ser6)-Goserelin is typically administered via subcutaneous injection and is known for its efficacy in managing hormone-dependent tumors and conditions. Its pharmacological profile includes a favorable safety and tolerability profile, although potential side effects may include hot flashes, decreased libido, and other hormonal-related symptoms.
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Found 3 products.