CAS 66504-75-4

Bicifadine hydrochloride

Description:

Bicifadine hydrochloride is a chemical compound that belongs to the class of analgesics, primarily used for its pain-relieving properties. It is characterized by its dual mechanism of action, which involves both opioid and non-opioid pathways, making it effective in managing moderate to severe pain. The compound is typically administered in its hydrochloride salt form, enhancing its solubility and bioavailability. Bicifadine has been studied for its potential benefits in treating various pain conditions, including postoperative pain and chronic pain syndromes. Its pharmacological profile suggests a lower risk of addiction compared to traditional opioids, although caution is still advised due to potential side effects such as gastrointestinal disturbances, dizziness, or sedation. As with any medication, the therapeutic use of Bicifadine hydrochloride should be guided by a healthcare professional, considering individual patient factors and potential drug interactions. Overall, Bicifadine hydrochloride represents a noteworthy option in the landscape of analgesic therapies, particularly for patients seeking alternatives to conventional opioid medications.

Formula: C₁₂H₁₅N·ClH

InChI: InChI=1S/C12H15N.ClH/c1-9-2-4-10(5-3-9)12-6-11(12)7-13-8-12;/h2-5,11,13H,6-8H2,1H3;1H

InChI key: InChIKey=OTZOPAFTLUOBOM-UHFFFAOYSA-N

SMILES: CC1=CC=C(C23C(C2)CNC3)C=C1.Cl

Synonyms:

• (±)-1-(4-Methylphenyl)-3-azabicyclo[3.1.0]hexane Hydrochloride
• (±)-1-p-Tolyl-3-azabicyclo[3.1.0]hexane Hydrochloride
• 3-Azabicyclo[3.1.0]hexane, 1-(4-methylphenyl)-, hydrochloride
• 3-Azabicyclo[3.1.0]hexane, 1-(4-methylphenyl)-, hydrochloride (1:1)
• Bicifadine hydrochloride
• Cl 220075
• Mcv 4147
• Nih 9542

Bicifadine Hydrochloride

Controlled Product

CAS: 66504-75-4

Applications Bicifadine Hydrochloride is a novel non-narcotic analgesic drug for the treatment of acute pain, chronic pain, and symptoms of neuropathic disorders.
References Wang, R., et al.: J. Clin. Pharmacol., 22, 160 (1982), Stephenson, G., et al.: Adv. Drug Delivery Rev., 48, 67 (2001), Blanco, M., et al.: J. Pharm. Sci., 92, 823 (2003), Woo, Y., et al.: J. Pharm. Biomed. Anal., 36, 955 (2005),

Formula: C₁₂H₁₅N·HCl

Color and Shape: Neat

Molecular weight: 173.26 + (36.46)

Ref: TR-B382250

Bicifadine hydrochloride

CAS: 66504-75-4

noradrenalin transporter antagonist

Formula: C₁₂H₁₆ClN

Purity: 98%

Color and Shape: Solid

Molecular weight: 209.715

Ref: TM-T22603