CAS 66722-44-9
:Bisoprolol
Description:
Bisoprolol is a selective beta-1 adrenergic antagonist, primarily used in the management of hypertension and heart failure. It belongs to the class of medications known as beta-blockers, which work by blocking the effects of adrenaline on the heart, leading to a decrease in heart rate and blood pressure. Chemically, bisoprolol is characterized by its structure, which includes a phenol ring and a side chain that contributes to its selectivity for beta-1 receptors. It is typically administered orally and has a relatively long half-life, allowing for once-daily dosing. Bisoprolol is well-absorbed in the gastrointestinal tract, with a bioavailability that can be influenced by first-pass metabolism. Common side effects may include fatigue, dizziness, and bradycardia, while contraindications include severe asthma and certain heart conditions. Overall, bisoprolol is an effective therapeutic agent for cardiovascular conditions, with a favorable safety profile when used appropriately.
Formula:C18H31NO4
InChI:InChI=1/C18H31NO4/c1-14(2)19-11-17(20)13-23-18-7-5-16(6-8-18)12-21-9-10-22-15(3)4/h5-8,14-15,17,19-20H,9-13H2,1-4H3
InChI key:InChIKey=VHYCDWMUTMEGQY-UHFFFAOYSA-N
SMILES:O(CC(CNC(C)C)O)C1=CC=C(COCCOC(C)C)C=C1
Synonyms:- 1-(Propan-2-ylamino)-3-[4-(2-propan-2-yloxyethoxymethyl)phenoxy]propan-2-ol
- 1-(p-2-Isopropoxyethoxymethylphenoxy)-3-isopropylaminopropan-2-ol
- 1-[4-(2-Isopropoxy-ethoxymethyl)-phenoxy]-3-isopropylamino-propan-2-ol
- 1-[4-[[2-(1-Methylethoxy)ethoxy]methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol
- 2-Propanol, 1-[4-[[2-(1-methylethoxy)ethoxy]methyl]phenoxy]-3-[(1-methylethyl)amino]-
- Bisoprolol
- Bisoprolol base
- Cardensiel
- Konkor
- Racemic Bisoprolol
- Ty 0201
- Bisoprolol(Hemifumalate)
- 1-[(1-Methylethyl)amino]-3-[4-[[2-(1-methylethoxy)ethoxy]methyl]phenoxy]-2-propanol
- 1-[4-[[2-(1-Methylethoxy)ethoxy]methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol-d5
- (R)-1-[(1-Methylethyl)amino]-3-[4-[[2-(1-methylethoxy)ethoxy]methyl]phenoxy]-2-propanol
- (R)-1-(Isopropylamino)-3-[4-(2-isopropoxyethoxymethyl)phenoxy]-2-propanol
- Bisoprolol-D5
- 1-[4-[2-(1-Methylethoxy)ethoxymethyl]phenoxy]-3-(1-methylethylamino)propan-2-ol
- Bisoprolo
- (S)-1-(Isopropylamino)-3-[4-(2-isopropoxyethoxymethyl)phenoxy]-2-propanol
- (S)-1-[(1-Methylethyl)amino]-3-[4-[[2-(1-methylethoxy)ethoxy]methyl]phenoxy]-2-propanol
- See more synonyms
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Found 7 products.
Bisoprolol Hemifumarate
CAS:Formula:C18H31NO4C4H4O4Purity:>98.0%(T)(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:383.49Bisoprolol
CAS:Controlled Product<p>Bisoprolol is a selective beta-adrenergic receptor antagonist that is used to treat high blood pressure and congestive heart failure. It also has a protective effect on the myocardium. Bisoprolol blocks the action of catecholamines on beta-2 receptors in the heart and peripheral vascular system, reducing heart rate, cardiac output, and blood pressure. This drug also inhibits calcium release from the sarcoplasmic reticulum of cardiac muscle cells by binding to the ryanodine receptor. Bisoprolol is not absorbed when taken orally, so it must be administered by injection or intravenously. The drug’s activity can be monitored using chromatographic analysis to measure levels of bisoprolol in human serum or blood pressure monitoring to measure changes in blood pressure after administration of bisoprolol.</p>Formula:C18H31NO4Purity:Min. 95%Color and Shape:PowderMolecular weight:325.44 g/mol
