CAS 668463-35-2

RPR-260243

Description:

RPR-260243, with the CAS number 668463-35-2, is a chemical compound that has garnered attention in pharmaceutical research, particularly for its potential therapeutic applications. It is classified as a selective inhibitor of certain enzymes, which may play a role in various biological processes. The compound exhibits a specific mechanism of action that targets particular pathways, making it a candidate for further investigation in the treatment of conditions such as inflammation or cancer. RPR-260243 is characterized by its unique molecular structure, which contributes to its biological activity and selectivity. Additionally, studies have indicated that it may possess favorable pharmacokinetic properties, including absorption, distribution, metabolism, and excretion profiles. However, detailed information regarding its safety, efficacy, and potential side effects is still under investigation, as it is primarily in the research phase. As with many compounds in development, further studies are necessary to fully understand its characteristics and therapeutic potential.

Formula: C₂₈H₂₅F₃N₂O₄

Synonyms:

• 100866
• (3R,4R)-4-[3-(6-Methoxyquinolin-4-yl)-3-oxo-propyl]-1-[3-(2,3,5-trifluoro-phenyl)-prop-2-ynyl]-piperidine-3-carboxylic acid
• (3R,4R)-4-[3-(6-Methoxyquinolin-4-yl)-3-oxo-propyl]-1-[3-(2,3,5-trifluoro-phenyl)-prop-2-ynyl]
• RPR-260243
• RPR 260243;RPR260243
• CS-2094
• 3-Piperidinecarboxylic acid, 4-[3-(6-methoxy-4-quinolinyl)-3-oxopropyl]-1-[3-(2,3,5-trifluorophenyl)-2-propyn-1-yl]-, (3R,4R)-

RPR-260243 

CAS: 668463-35-2

Formula: C₂₈H₂₅F₃N₂O₄

Purity: 99.37%

Molecular weight: 510.5043

Ref: IN-DA00FC1R

RPR-260243

CAS: 668463-35-2

RPR-260243 is a chemical compound that is a potassium ion channel blocker. This drug blocks the voltage-gated potassium channels and prevents the flow of potassium ions in cardiac tissues, thereby blocking the propagation of an action potential. The affinity values for RPR-260243 have been determined using binding studies on rat heart tissue and human recombinant cardiac channels. The molecular modeling studies show that RPR-260243 binds to the channel of potassium ions through hydrogen bonding interactions with Arg45, Lys53, and Asp52.

Formula: C₂₈H₂₅F₃N₂O₄

Purity: Min. 95%

Molecular weight: 510.5 g/mol

Ref: 3D-TBB46335

RPR-260243

CAS: 668463-35-2

RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).

Formula: C₂₈H₂₅F₃N₂O₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 510.5

Ref: TM-T16796