CAS 7085-45-2

Biperiden lactate

Description:

Biperiden lactate is a chemical compound primarily used in the treatment of Parkinson's disease and other movement disorders. It acts as an anticholinergic agent, helping to alleviate symptoms such as tremors and rigidity by blocking the action of acetylcholine in the central nervous system. The compound is a lactate salt of biperiden, which enhances its solubility and bioavailability. Biperiden itself is a piperidine derivative, characterized by its ability to cross the blood-brain barrier, making it effective for neurological applications. In terms of physical properties, biperiden lactate is typically a white to off-white crystalline powder, and it is soluble in water and alcohol. Its pharmacological profile includes side effects such as dry mouth, blurred vision, and constipation, which are common among anticholinergic medications. As with any medication, it is essential to use biperiden lactate under medical supervision to manage dosage and monitor for potential adverse effects.

Formula: C₂₁H₂₉NO·C₃H₆O₃

InChI: InChI=1S/C21H29NO.C3H6O3/c23-21(19-7-3-1-4-8-19,11-14-22-12-5-2-6-13-22)20-16-17-9-10-18(20)15-17;1-2(4)3(5)6/h1,3-4,7-10,17-18,20,23H,2,5-6,11-16H2;2,4H,1H3,(H,5,6)

InChI key: InChIKey=GLPUBCPQWZZFNJ-UHFFFAOYSA-N

SMILES: C(CCN1CCCCC1)(O)(C2C3CC(C2)C=C3)C4=CC=CC=C4.C(C(O)=O)(C)O

Synonyms:

• 1-Piperidinepropanol, alpha-bicyclo(2.2.1)hept-5-en-2-yl-alpha-phenyl-, compd. with 2-hydroxypropanoic acid (1:1)
• 1-Piperidinepropanol, α-5-norbornen-2-yl-α-phenyl-, lactate
• 1-Piperidinepropanol, α-bicyclo[2.2.1]hept-5-en-2-yl-α-phenyl-, 2-hydroxypropanoate (salt)
• 2-Hydroxypropanoic Acid - 1-(Bicyclo[2.2.1]Hept-5-En-2-Yl)-1-Phenyl-3-(Piperidin-1-Yl)Propan-1-Ol (1:1)
• Akineton
• Akineton Lactate
• Biperiden lactate [USAN:BAN:JAN]
• Lactic acid, compd. with alpha-5-norbornen-2-yl-alpha-phenyl-1-piperidinepropanol (1:1)
• Lactic acid, compd. with α-5-norbornen-2-yl-α-phenyl-1-piperidinepropanol (1:1)
• Lactic acid, compound with alpha-bicyclo(2.2.1)hept-5-en-2-yl-alpha-phenylpiperidin-1-propanol (1:1)
• Propanoic acid, 2-hydroxy-, compd. with α-bicyclo[2.2.1]hept-5-en-2-yl-α-phenyl-1-piperidinepropanol (1:1)
• Unii-09Td6C5147
• alpha-5-Norbornen-2-yl-alpha-phenyl-1-piperidinepropanol compd. with lactic acid (1:1)
• alpha-5-Norbornen-2-yl-alpha-phenyl-1-piperidinepropanol lactate (salt)
• α-(Bicyclo[2.2.1]hept-5-en-2-yl)-α-phenyl-1-piperidine propanol lactate

Biperiden lactate

CAS: 7085-45-2

Biperiden lactate is a biochemical.

Formula: C₂₄H₃₅NO₄

Color and Shape: Solid

Molecular weight: 401.54

Ref: TM-T30456

Biperiden Lactate

Controlled Product

CAS: 7085-45-2

Applications Biperiden Lactate is antiparkinsonian; non-selective muscarinic receptor antagonist. Biperiden is used for the adjunctive treatment of all forms of Parkinson′s Disease (postencephalitic, idiopathic, and arteriosclerotic); also commonly used to improve parkinsonian signs and symptoms related to antipsychotic drug therapy.
References Patela, Y., et al.: Talanta, 47, 625 (1998), Bebawy, L., et al: J. Pharm. Biomed. Anal., 20, 663 (1999), Dinc, E., et al.: J. Pharm. Biomed. Anal., 28, 591 (2002),

Formula: C₂₁H₂₉NO·C₃H₆O₃

Color and Shape: Neat

Molecular weight: 311.46 + (90.08)

Ref: TR-B397843