CAS 7125-67-9

metoquizine

Description:

Metoquizine is a chemical compound classified as an antihistamine and is primarily used for its antiemetic properties, particularly in the treatment of motion sickness and nausea. It functions by blocking histamine receptors, which helps alleviate symptoms associated with these conditions. Metoquizine is known for its ability to cross the blood-brain barrier, which contributes to its effectiveness in managing central nervous system-related symptoms. The compound typically exhibits a moderate to high solubility in organic solvents, while its solubility in water can vary. Its pharmacological profile includes sedative effects, which may limit its use in certain populations or situations. As with many medications, potential side effects can include drowsiness, dry mouth, and dizziness. Metoquizine's safety and efficacy have been evaluated in various clinical settings, and it is important for users to follow prescribed dosages to minimize adverse effects. Overall, metoquizine represents a valuable option in the pharmacological management of nausea and motion sickness.

Formula: C₂₂H₂₇N₅O

InChI: InChI=1/C22H27N5O/c1-13-8-14(2)27(24-13)22(28)23-16-10-18-17-6-5-7-19-21(17)15(11-25(19)3)9-20(18)26(4)12-16/h5-8,11,16,18,20H,9-10,12H2,1-4H3,(H,23,28)/t16-,18-,20-/m1/s1

Synonyms:

• Metoquizinum
• UNII-2DW6SEL94L
• Metoquizine
• 3,5-Dimethyl-N-(4,6,6a,7,8,9,10,10a-octahydro-4,7-dimethylindolo(4,3-fg)-9-yl)pyrazole-1-carboxamide
• 3,5-Dimethyl-N-(4,6,6a,7,8,9,10,10a-octahydro-4,7-dimethyl-indolol(4,3-f,g)chinolin-9-yl)pyrazol-1-carboxamid
• N-(1,6-Dimethyl-8beta-ergolinyl)-3,5-dimethyl-1-pyrazolcarboxamid
• Metoquizine [USAN:INN]
• 1H-Pyrazole-1-carboxamide, 3,5-dimethyl-N-(4,6,6a,7,8,9,10,10a-octahydro-4,7-dimethylindolo(4,3-fg)quinolin-9-yl)
• Ly 42406
• N-[(8beta)-1,6-dimethylergolin-8-yl]-3,5-dimethyl-1H-pyrazole-1-carboxamide
• Lilly 42406
• 3,5-Dimethyl-N-(4,6,6a,7,8,9,10,10a-octahydro-4,7-dimethylindolo(4,3-fg)quinolin-9-yl)pyrazole-1-carboxamide

Metoquizine

CAS: 7125-67-9

Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.

Formula: C₂₂H₂₇N₅O

Purity: 98%

Color and Shape: Solid

Molecular weight: 377.48

Ref: TM-T25805