CAS 72522-13-5
:(-)-Eptazocine
Description:
(-)-Eptazocine is a synthetic opioid analgesic that belongs to the class of benzomorphan derivatives. It is primarily characterized by its potent analgesic properties, which are attributed to its action as a mixed agonist-antagonist at opioid receptors, particularly the mu and kappa receptors. This dual action allows it to provide pain relief while potentially minimizing some of the side effects commonly associated with pure opioid agonists, such as respiratory depression. (-)-Eptazocine is known for its relatively low potential for abuse compared to traditional opioids, making it a subject of interest in pain management. The compound is typically administered in a clinical setting and has been studied for its efficacy in treating moderate to severe pain. Its chemical structure includes a complex arrangement of rings and functional groups that contribute to its pharmacological activity. As with all opioids, careful consideration of dosage and monitoring for side effects is essential in its use.
Formula:C15H21NO
InChI:InChI=1S/C15H21NO/c1-15-5-6-16(2)10-11(9-15)7-12-3-4-13(17)8-14(12)15/h3-4,8,11,17H,5-7,9-10H2,1-2H3/t11?,15-/m1/s1
InChI key:InChIKey=ZOWQTJXNFTWSCS-JOPIAHFSSA-N
SMILES:C[C@]12C=3C(CC(C1)(CN(C)CC2)[H])=CC=C(O)C3
Synonyms:- (-)-1,4-Dimethyl-10-hydroxy-2,3,4,5,6,7-hexahydro-1,6-methano-1H-4-benzazonine
- (1S,6S)-1,4-dimethyl-2,3,4,5,6,7-hexahydro-1H-1,6-methano-4-benzazonin-10-ol
- (1S,6S)-2,3,4,5,6,7-Hexahydro-1,4-dimethyl-1,6-methano-1H-4-benzazonin-10-ol
- 1,4-dimethyl-2,3,4,5,6,7-hexahydro-1H-1,6-methano-4-benzazonin-10-ol
- 1,6-Methano-1H-4-benzazonin-10-ol, 2,3,4,5,6,7-hexahydro-1,4-dimethyl-, (1S)-
- 1,6-Methano-1H-4-benzazonin-10-ol, 2,3,4,5,6,7-hexahydro-1,4-dimethyl-, (1S,6S)-
- Sedapain
- Eptazocine
- (-)-Eptazocine
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Found 4 products.
Eptazocine
CAS:Eptazocine is a peptide that belongs to the group of activators. It is used as a research tool in cell biology, pharmacology, and other life science fields. Eptazocine has been shown to inhibit the activity of ion channels and receptors. Furthermore, it has been used as an antibody to study protein interactions. Eptazocine can be used as a reagent for studying ligand-receptor interactions and is a member of the opioid receptor family. It binds to alpha-subunits of opioid receptors, which are G protein-coupled receptors that activate phospholipase C and inhibit adenylyl cyclase.
Formula:C15H21NOPurity:Min. 95%Molecular weight:231.33 g/mol
