CAS 75644-90-5
:(D-ser2)-leucine enkephalin-thr acetate
Description:
(D-ser2)-leucine enkephalin-thr acetate, with the CAS number 75644-90-5, is a synthetic peptide that belongs to the class of enkephalins, which are endogenous opioid peptides. This compound is characterized by its specific amino acid sequence, which includes D-serine and leucine, contributing to its biological activity. It functions primarily as a neurotransmitter and neuromodulator, interacting with opioid receptors in the central nervous system to produce analgesic effects. The acetate group in its structure enhances its solubility and stability, making it suitable for various biochemical applications. As a peptide, it is typically synthesized through solid-phase peptide synthesis techniques and may exhibit properties such as high specificity for certain receptors, potential for therapeutic use in pain management, and modulation of mood and stress responses. Its stability, bioavailability, and pharmacokinetic properties are critical for its effectiveness in research and potential clinical applications.
Formula:C33H46N6O10
InChI:InChI=1/C33H46N6O10/c1-18(2)13-24(32(47)39-28(19(3)41)33(48)49)37-31(46)25(15-20-7-5-4-6-8-20)36-27(43)16-35-30(45)26(17-40)38-29(44)23(34)14-21-9-11-22(42)12-10-21/h4-12,18-19,23-26,28,40-42H,13-17,34H2,1-3H3,(H,35,45)(H,36,43)(H,37,46)(H,38,44)(H,39,47)(H,48,49)/t19-,23+,24+,25+,26-,28+/m1/s1
Synonyms:- Enkephalin, Ser(2), Leu(5), Thr(6)-
- 2-Ser-thr-leu-enkephalin
- Dslet
- Dstle
- Dislet
- Enkephalin-leu, ser(2)-thr-
- Enkephalin-leu, seryl(2)-threonine-
- Leu-enkephalin, ser(2)-thr-
- Leucine-enkephalin, ser(2)-thr-
- Ser(2)-leu(5)-enkephalin-thr(6)
- Tyr-ser-gly-phe-leu-thr
- Tyrosyl-seryl-glycyl-phenylalanyl-leucyl-threonine
- L-Threonine, L-tyrosyl-D-serylglycyl-L-phenylalanyl-L-leucyl-
- L-Threonine, N-(N-(N-(N-(N-L-tyrosyl-D-seryl)glycyl)-L-phenylalanyl)-L-leucyl)-
- See more synonyms
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100
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90
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Found 2 products.
(D-Ser2)-Leu-Enkephalin-Thr
CAS:(D-Ser2)-Leu-Enkephalin-Thr H-Tyr-D-Ser-Gly-Phe-Leu-Thr-OH is a cyclic peptide that has been shown to activate the κ-opioid receptor. The peptide has been used in studies of the intracellular calcium concentration and glomerular filtration rate in kidney cells, as well as the antinociceptive effects of opioid drugs on mice. This drug has also been shown to have effects on cyclic AMP levels and α 1 -adrenergic receptors in neuro2a cells.Formula:C33H46N6O10Purity:Min. 95%Color and Shape:SolidMolecular weight:686.75 g/mol

