CAS 75696-02-5
:Cinolazepam
Description:
Cinolazepam is a benzodiazepine derivative primarily used for its anxiolytic, sedative, and muscle relaxant properties. It is characterized by its ability to enhance the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased neuronal inhibition. This mechanism contributes to its therapeutic effects in treating anxiety disorders and sleep disturbances. Cinolazepam is typically administered orally and has a relatively long half-life, which can result in prolonged effects. The substance is known for its low potential for abuse compared to other benzodiazepines, although caution is advised due to the risk of dependence with prolonged use. Common side effects may include drowsiness, dizziness, and cognitive impairment. As with other medications in its class, it is essential to use cinolazepam under medical supervision to mitigate risks and ensure appropriate dosing. Its chemical structure includes a diazepine ring, which is characteristic of benzodiazepines, contributing to its pharmacological profile.
Formula:C18H13ClFN3O2
InChI:InChI=1S/C18H13ClFN3O2/c19-11-6-7-15-13(10-11)16(12-4-1-2-5-14(12)20)22-17(24)18(25)23(15)9-3-8-21/h1-2,4-7,10,17,24H,3,9H2
InChI key:InChIKey=XAXMYHMKTCNRRZ-UHFFFAOYSA-N
SMILES:C(CC#N)N1C=2C(C(=NC(O)C1=O)C3=C(F)C=CC=C3)=CC(Cl)=CC2
Synonyms:- 1H-1,4-Benzodiazepine-1-propanenitrile, 2,3-dihydro-7-chloro-5-(2-fluorophenyl)-2-oxo-
- 1H-1,4-Benzodiazepine-1-propanenitrile, 7-chloro-5-(2-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-
- 3-[7-chloro-5-(2-fluorophenyl)-3-hydroxy-2-oxo-2,3-dihydro-1H-1,4-benzodiazepin-1-yl]propanenitrile
- 7-Chloro-5-(2-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-1H-1,4-benzodiazepine-1-propanenitrile
- 7-Chloro-5-(o-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-1H-1,4-benzodiazepine-1-propionitrile
- Brn 5359831
- Cinolazepam [INN]
- Cinolazepamum
- Cinolazepamum [INN-Latin]
- Gerodorm
- Ox 373
- Unii-68P0556B0U
- See more synonyms
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Found 3 products.
Cinolazepam
CAS:Cinolazepam is a benzodiazepine derivative drug.It has a powerful sedative effect, so it is mainly used as a hypnotic.Formula:C18H13ClFN3O2Color and Shape:SolidMolecular weight:357.77Cinolazepam
CAS:Controlled ProductCinolazepam is a benzodiazepine derivative, which is a synthetic product that acts primarily as a central nervous system depressant. Its mode of action involves enhancing the effect of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, resulting in increased inhibitory effects and neuronal hyperpolarization. This leads to its characteristic sedative and anxiolytic properties.Cinolazepam is utilized in therapeutic settings primarily as a hypnotic for the management of insomnia, particularly in cases involving difficulty in sleep initiation. It may also offer anxiolytic benefits, although it is less commonly prescribed for generalized anxiety disorders compared to other benzodiazepines. Its pharmacokinetic profile includes a relatively short half-life, favoring its use as a sleep aid with reduced risk of next-day residual effects. However, caution is warranted due to the potential for tolerance, dependence, and withdrawal phenomena typical of benzodiazepines. Therefore, its use is recommended for short-term treatment periods under strict medical supervision.Formula:C18H13ClFN3O2Purity:Min. 95%Molecular weight:357.8 g/mol


