CAS 77862-92-1

Falipamil

Description:

Falipamil, with the CAS number 77862-92-1, is a chemical compound that belongs to the class of calcium channel blockers. It is primarily used in the medical field for its antihypertensive properties, helping to manage high blood pressure and certain types of angina. The compound works by inhibiting the influx of calcium ions through voltage-gated calcium channels in cardiac and smooth muscle cells, leading to vasodilation and reduced myocardial contractility. This mechanism helps to lower blood pressure and improve blood flow. Falipamil is characterized by its specific molecular structure, which contributes to its pharmacological activity. It is typically administered in a controlled dosage to ensure efficacy while minimizing potential side effects, which may include dizziness, headache, or gastrointestinal disturbances. As with many pharmaceuticals, the safety and effectiveness of Falipamil are evaluated through clinical trials, and it is important for patients to follow medical advice when using this medication.

Formula: C₂₄H₃₂N₂O₅

InChI: InChI=1/C24H32N2O5/c1-25(12-9-17-7-8-20(28-2)21(13-17)29-3)10-6-11-26-16-18-14-22(30-4)23(31-5)15-19(18)24(26)27/h7-8,13-15H,6,9-12,16H2,1-5H3

InChI key: InChIKey=UUMGNNQOCVDZDG-UHFFFAOYSA-N

SMILES: O=C1C=2C(CN1CCCN(CCC3=CC(OC)=C(OC)C=C3)C)=CC(OC)=C(OC)C2

Synonyms:

• 1H-Isoindol-1-one, 2-(3-((2-(3,4-dimethoxyphenyl)ethyl)methylamino)propyl)-2,3-dihydro-5,6-dimethoxy-
• 2-(3-((3,4-Dimethoxyphenetyl)methylamino)propyl)-5,6-dimethoxyphthalimidine
• 2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}propyl)-5,6-dimethoxy-2,3-dihydro-1H-isoindol-1-one
• 2-[3-[[2-(3,4-Dimethoxyphenyl)ethyl]methylamino]propyl]-2,3-dihydro-5,6-dimethoxy-1H-isoindol-1-one
• Aq-A 39
• Falipamil [INN]
• Falipamilum
• Falipamilum [INN-Latin]
• Unii-N6A93Zmn7U
• Falipamil
• 2-[3-[2-(3,4-Dimethoxyphenyl)ethyl(methyl)amino]propyl]-2,3-dihydro-5,6-dimethoxy-1H-isoindol-1-one

Falipamil

Controlled Product

CAS: 77862-92-1

Applications Falipamil is a specific bradycardic agent and a calcium channel blocker.
References Boucher, M., et al.: Eur. J. Pharmacol., 306, 93 (1996), Mubagwa, K., et al.: Arch. Int. Pharmacodyn. Ther., 286, 71 (1987), Chaudhry, A., et al.: Development Cardiovascular Medicine, 46, 196 (1985), Ogiwara, Y., et al.: Jpn Heart J., 29, (1988)

Formula: C₂₄H₃₂N₂O₅

Color and Shape: Neat

Molecular weight: 428.52

Ref: TR-F101116

Falipamil

CAS: 77862-92-1

Falipamil is a peptide that inhibits the interaction of proteins. It binds to the receptor site of the protein and blocks its activity. Falipamil is not an agonist, meaning it does not activate the receptor. It is also a ligand, which means it binds to specific receptors and activates them. Falipamil has been shown to be an excellent research tool for studying protein interactions, as well as being used in antibody production. This product can be used for life science research and has high purity with a CAS Number of 77862-92-1.

Formula: C₂₄H₃₂N₂O₅

Purity: Min. 95%

Molecular weight: 428.5 g/mol

Ref: 3D-CDA86292

Falipamil

CAS: 77862-92-1

Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.

Formula: C₂₄H₃₂N₂O₅

Purity: 98%

Color and Shape: Solid

Molecular weight: 428.52

Ref: TM-T27302