CAS 78-44-4

Carisoprodol

Description:

Carisoprodol is a centrally acting muscle relaxant commonly used to relieve muscle pain and discomfort associated with acute musculoskeletal conditions. It is classified as a carbamate derivative and functions primarily by interrupting neuronal communication within the reticular formation and spinal cord, leading to sedation and muscle relaxation. The substance is typically administered orally and is known for its rapid onset of action. Carisoprodol is metabolized in the liver to its active metabolite, meprobamate, which contributes to its sedative effects. The chemical formula for carisoprodol is C12H24N2O4S, and it has a molecular weight of approximately 256.39 g/mol. It is generally well-absorbed from the gastrointestinal tract, but its use is associated with potential side effects, including drowsiness, dizziness, and dependence, particularly with prolonged use. Due to these risks, carisoprodol is classified as a controlled substance in several jurisdictions, necessitating careful prescribing and monitoring by healthcare professionals.

Formula: C₁₂H₂₄N₂O₄

InChI: InChI=1S/C12H24N2O4/c1-5-6-12(4,7-17-10(13)15)8-18-11(16)14-9(2)3/h9H,5-8H2,1-4H3,(H2,13,15)(H,14,16)

InChI key: InChIKey=OFZCIYFFPZCNJE-UHFFFAOYSA-N

SMILES: C(COC(NC(C)C)=O)(COC(N)=O)(CCC)C

Synonyms:

• 2-Carbamoyloxymethyl-2-methylpentyl isopropylcarbamate
• 2-Methyl-2-propyl-1,3-propanediol carbamate isopropylcarbamate
• Apesan
• Arusal
• Atonalyt
• Calenfa
• Caprodat
• Carbamic acid, N-(1-methylethyl)-, 2-[[(aminocarbonyl)oxy]methyl]-2-methylpentyl ester
• Carbamic acid, isopropyl-, 2-(hydroxymethyl)-2-methylpentyl ester carbamate (ester)
• Carbamic acid, isopropyl-, 2-(hydroxymethyl)-2-methylpentyl ester, carbamate
• Carisol
• Carisoma
• Carisoprodate
• Carisoprodatum
• Carisoprodol
• Domarax
• Flexal
• Flexartal
• Isobamate
• Isomeprobamate
• Isopropyl meprobamate
• Isoprotan
• Isoprotane
• Isoprothane
• Izoprotan
• Miolisodal
• Mioril
• N-Isopropyl-2-methyl-2-propyl-1,3-propanediol dicarbamate
• Nih 10966
• Nsc 172124
• Rela
• Rela (carbamic acid)
• Relasom
• Sanoma
• Skutamil
• Soma
• Somadril
• Somalgit
• Stialgin

Carisoprodol

CAS: 78-44-4

Formula: C₁₂H₂₄N₂O₄

Purity: >98.0%(HPLC)(N)

Color and Shape: White to Almost white powder to crystal

Molecular weight: 260.33

Ref: 3B-C3573

Carisoprodol, 1mg/ml in Methanol

CAS: 78-44-4

Color and Shape: Single Solution

Ref: LP-CSP-1101-1LM

Carisoprodol

Controlled Product

CAS: 78-44-4

Color and Shape: Neat

Ref: LP-CSP-1101-10

Carisoprodol 1.0 mg/ml in Methanol

CAS: 78-44-4

Color and Shape: Single Solution

Ref: 61-AMP0782.00-01

Carisoprodol

CAS: 78-44-4

Formula: C₁₂H₂₄N₂O₄

Purity: ≥ 98.0%

Color and Shape: White to almost white crystalline powder

Molecular weight: 260.33

Ref: 7W-GP0362

Carisoprodol

Controlled Product

CAS: 78-44-4

Formula: C₁₂H₂₄N₂O₄

Color and Shape: Neat

Molecular weight: 260.33

Ref: 86-MM0782.00

Carisoprodol

CAS: 78-44-4

Color and Shape: Neat

Ref: 61-FOR0782.00

Carisoprodol

Controlled Product

CAS: 78-44-4

Applications Muscle relaxant (skeletal).
References Musso, D., et al.: J. Med. Chem. 46, 399 (2003), Newman, P., et al.: Eur. J. Clin. Pharm., 23, 31 (1982).

Formula: C₁₂H₂₄N₂O₄

Color and Shape: White To Off-White

Molecular weight: 260.33

Ref: TR-C183580

Carisoprodol

Controlled Product

CAS: 78-44-4

Carisoprodol is a synthetic compound that is used as a reaction component, reagent, and useful scaffold in the synthesis of pharmaceuticals. Carisoprodol has been shown to be a high-quality research chemical with versatile building blocks. It can be used as an intermediate in the synthesis of complex compounds such as anticonvulsants and muscle relaxants. Carisoprodol is also a fine chemical with CAS number 78-44-4.

Formula: C₁₂H₂₄N₂O₄

Purity: Min. 98 Area-%

Molecular weight: 260.33 g/mol

Ref: 3D-W-104280

2-Methyl-2-propyl-1,3-propanediol carbamate isopropylcarbamate

Controlled Product

CAS: 78-44-4

2-Methyl-2-propyl-1,3-propanediol carbamate isopropylcarbamate (2MPPC) is a prodrug that is metabolized to carisoprodol. It has been shown to have a high affinity for the neuronal death receptor, TNFRSF25, and can cause neuronal death in vitro. In vivo studies show that 2MPPC causes axonal growth and promotes locomotor activity. 2MPPC also inhibits the production of prostaglandin E2 and nitric oxide, which may be due to its inhibition of cyclooxygenase 1 and nitric oxide synthase 1. Clinical pathology studies reveal that 2MPPC does not cause toxicity at therapeutic doses. Histological analysis shows that 2MPPC does not affect the granule neurons in the dentate gyrus region of the hippocampus.

Formula: C₁₂H₂₄N₂O₄

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 260.33 g/mol

Ref: 3D-FM19816

Carisoprodol (1 mg/ml in Methanol)

Controlled Product

CAS: 78-44-4

Formula: C₁₂H₂₄N₂O₄

Color and Shape: Colourless

Molecular weight: 260.33

Ref: TR-KIT2020

Carisoprodol CIV

Controlled Product

CAS: 78-44-4

Acyclic amides (including acyclic carbamates) and their derivatives and salts thereof, nesoi

Formula: C₁₂H₂₄N₂O₄

Color and Shape: White Powder

Molecular weight: 260.17361

Ref: 45-1096600

Carisoprodol

Controlled Product

CAS: 78-44-4

Formula: C₁₂H₂₄N₂O₄

Color and Shape: Neat

Molecular weight: 260.33

Ref: 04-C11043500