CAS 786686-79-1

2-methyl-4-[4-(trideuteriomethyl)piperazin-1-yl]-10H-thieno[2,3-b][1,5]benzodiazepine

Description:

2-Methyl-4-[4-(trideuteriomethyl)piperazin-1-yl]-10H-thieno[2,3-b][1,5]benzodiazepine is a synthetic compound belonging to the benzodiazepine class, characterized by its complex structure that includes a thieno[2,3-b][1,5]benzodiazepine core. This compound features a methyl group at the 2-position and a piperazine ring substituted at the 4-position with a trideuteriomethyl group, which indicates the presence of deuterium isotopes in the methyl group. The presence of deuterium can influence the compound's pharmacokinetics and metabolic stability. Typically, benzodiazepines exhibit anxiolytic, sedative, and muscle relaxant properties, and their activity is often mediated through interactions with the GABA-A receptor. The specific characteristics of this compound, including its solubility, stability, and biological activity, would depend on its molecular structure and the presence of functional groups. As a research chemical, it may be of interest in pharmacological studies, particularly in understanding the effects of isotopic substitution on drug behavior.

Formula: C₁₇H₁₇D₃N₄S

InChI: InChI=1/C17H20N4S/c1-12-11-13-16(21-9-7-20(2)8-10-21)18-14-5-3-4-6-15(14)19-17(13)22-12/h3-6,11,19H,7-10H2,1-2H3/i2D3

SMILES: Cc1cc2C(=Nc3ccccc3Nc2s1)N1CCN(C([2H])([2H])[2H])CC1

Olanzapine-D3 1.0 mg/ml in Acetonitrile

CAS: 786686-79-1

Color and Shape: Single Solution

Ref: 61-AMP0329.81-11

Olanzapine-d3

CAS: 786686-79-1

Formula: C₁₇H₁₇D₃N₄S

Color and Shape: Yellow Solid

Molecular weight: 315.45

Ref: 4Z-O-012

Olanzapine-d3 (4-methyl-d3-piperazinyl)

CAS: 786686-79-1

Purity: 99 atom % D

Color and Shape: Yellow Solid

Molecular weight: 315.45

Ref: 3U-D7477

Olanzapine D3

CAS: 786686-79-1

Olanzapine D3 is the deuterium labeled Olanzapine.

Formula: C₁₇H₂₀N₄S

Purity: 98%

Color and Shape: Solid

Molecular weight: 315.45

Ref: TM-T12291

Olanzapine Impurity 35

CAS: 786686-79-1

Formula: C₆H₆N₂S

Color and Shape: Yellow Solid

Molecular weight: 138.19

Ref: 4Z-O-0120

Olanzapine-d3

Controlled Product

CAS: 786686-79-1

Applications Deuterated Olanzapine, a serotonin (5-HT2) and dopamine (D1/D2) receptor antagonist with anticholinergic activity. Antipsychotic.
References Moore, N.A., et al.: Curr. Opin Invest. Drugs, 2, 281 (1993), Baldwin, D.S. and Montgomery, S.A.: Int. Clin. Psychopharmacol., 10, 239 (1995), Tohen, M., et al.: Am. J. Psychiatry, 156, 702 (1999)

Formula: C₁₇₂H₃H₁₇N₄S

Color and Shape: Yellow To Brown

Molecular weight: 315.45

Ref: TR-O253752

Olanzapine-d3 (1 mg/ml in Acetonitrile)

Controlled Product

CAS: 786686-79-1

Formula: C₁₇₂H₃H₁₇N₄S

Color and Shape: Colourless

Molecular weight: 315.45

Ref: TR-KIT1635

Olanzapine d3

Controlled Product

CAS: 786686-79-1

Olanzapine d3 is a potent inhibitor of cancer cell growth and tumor formation. It works by inhibiting the activity of kinases, which are enzymes that play a key role in regulating the cell cycle. Olanzapine d3 has been shown to be effective against various types of cancer, including leukemia and solid tumors. This medicinal compound has anticancer properties due to its ability to induce apoptosis, or programmed cell death, in cancer cells. In addition, Olanzapine d3 has been used in Chinese medicine for its protein kinase inhibitory effects and is commonly found in urine samples as a result of metabolism. Overall, this compound shows great promise as an effective treatment option for those suffering from various forms of cancer.

Formula: C₁₇H₂₀N₄S

Purity: Min. 95%

Molecular weight: 315.5 g/mol

Ref: 3D-LGB68679