CAS 78715-23-8

Norbuprenorphine

Description:

Norbuprenorphine is a semi-synthetic opioid derived from buprenorphine, primarily known for its role as a metabolite of buprenorphine in the human body. It exhibits analgesic properties and interacts with the opioid receptors in the central nervous system, specifically the mu-opioid receptor, albeit with a lower affinity compared to its parent compound. Norbuprenorphine is characterized by its ability to act as a partial agonist, which means it can activate opioid receptors but to a lesser extent than full agonists, potentially leading to a reduced risk of respiratory depression. This compound is often studied for its implications in pain management and opioid dependence treatment. In terms of physical properties, norbuprenorphine is typically a white to off-white solid, and it is soluble in organic solvents but has limited solubility in water. Its pharmacokinetics and dynamics are of significant interest in both clinical and research settings, particularly regarding its role in opioid metabolism and its potential therapeutic applications.

Formula:C₂₅H₃₅NO₄

InChI:InChI=1S/C25H35NO4/c1-21(2,3)22(4,28)16-13-23-8-9-25(16,29-5)20-24(23)10-11-26-17(23)12-14-6-7-15(27)19(30-20)18(14)24/h6-7,16-17,20,26-28H,8-13H2,1-5H3/t16-,17-,20-,22+,23-,24+,25-/m1/s1

InChI key:InChIKey=YOYLLRBMGQRFTN-IOMBULRVSA-N

SMILES:O(C)[C@@]12[C@]3([C@@]45[C@@]([C@@](CC6=C4C(O3)=C(O)C=C6)(NCC5)[H])(C[C@@]1([C@]([C@](C)(C)C)(C)O)[H])CC2)[H]

Synonyms:

N-De(cyclopropylmethyl)buprenorphine
6,14-Ethenomorphinan-7-methanol, α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, (αS,5α,7α)-
Norbuprenorphine
6,14-Ethenomorphinan-7-methanol, α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, [5α,7α(S)]-
(αS,5α,7α)-α-(1,1-Dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-6,14-ethenomorphinan-7-methanol

Found 10 products.

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Norbuprenorphine
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Neat
Molecular weight:413.55
Ref: LP-BUP-982-FB
10mg
519.00€
VAT not included
50mg
1,973.00€
VAT not included
100mg
3,356.00€
VAT not included
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Norbuprenorphine 0.1 mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Colourless
Molecular weight:413.55
Ref: 61-AMP0120.10-02
1ml
92.00€
VAT not included
+ Info
Norbuprenorphine
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:White To Brown
Molecular weight:413.55
Ref: 61-FOR0120.10
5mg
340.00€
VAT not included
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Norbuprenorphine, 1mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Single Solution
Molecular weight:413.55
Ref: LP-BUP-982-FB-1LM
1ml
299.00€
VAT not included
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Norbuprenorphine 1.0 mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Colourless
Molecular weight:413.55
Ref: 61-AMP0120.10-01
1ml
626.00€
VAT not included
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(2S)-2-(4,5alpha-Epoxy-3-hydroxy-6-methoxy-6alpha,14-ethano-14alpha-morphinan-7alpha-yl)-3,3-dimethylbutan-2-ol (Norbuprenorphine)
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Neat
Molecular weight:413.55
Ref: 86-MM0120.10
25mg
2,091.00€
VAT not included
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Norbuprenorphine, 0.1mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Single Solution
Molecular weight:413.55
Ref: LP-BUP-982-FB-0.1LM
1ml
51.00€
VAT not included
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Norbuprenorphine
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Neat
Molecular weight:413.55
Ref: TR-N661300
1mg
188.00€
VAT not included
5mg
736.00€
VAT not included
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Norbuprenorphine (1.0 mg/mL in Methanol)
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Formula:C₂₅H₃₅NO₄
Color and Shape:Single Solution
Molecular weight:413.55
Ref: TR-KIT0695
1x1ml
946.00€
VAT not included
+ Info
Norbuprenorphine
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 78715-23-8
Please enquire for more information about Norbuprenorphine including the price, delivery time and more detailed product information at the technical inquiry form on this page
Formula:C₂₅H₃₅NO₄
Purity:Min. 95%
Molecular weight:413.55 g/mol
Ref: 3D-FN26431
5mg
Discontinued
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1g
Discontinued
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10mg
Discontinued
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Discontinued product