CAS 80012-43-7

Epinastine

Description:

Epinastine is an antihistamine primarily used for the treatment of allergic conjunctivitis and other allergic reactions. It functions as a selective H1 receptor antagonist, effectively blocking the action of histamine, a compound involved in allergic responses. Epinastine is characterized by its ability to alleviate symptoms such as itching, redness, and swelling associated with allergies. The substance is typically administered in the form of eye drops, allowing for localized treatment with minimal systemic absorption. Its chemical structure includes a piperidine ring, contributing to its pharmacological properties. Epinastine exhibits a favorable safety profile, with common side effects being mild and transient. Additionally, it has been noted for its dual action as both an antihistamine and a mast cell stabilizer, which helps prevent the release of histamine and other inflammatory mediators. Overall, Epinastine is an effective therapeutic option for managing allergic symptoms, particularly in ocular applications.

Formula: C₁₆H₁₅N₃

InChI: InChI=1S/C16H15N3/c17-16-18-10-15-13-7-3-1-5-11(13)9-12-6-2-4-8-14(12)19(15)16/h1-8,15H,9-10H2,(H2,17,18)

InChI key: InChIKey=WHWZLSFABNNENI-UHFFFAOYSA-N

SMILES: NC=1N2C(C=3C(CC=4C2=CC=CC4)=CC=CC3)CN1

Synonyms:

• 1H-Dibenz[c,f]imidazo[1,5-a]azepin-3-amine, 9,13b-dihydro-
• 3-Amino-9,13B-Dihydro-1H-Dibenz[C,F]Imidazo[1,5-A]Azepine
• 9,13b-Dihydro-1H-dibenz[c,f]imidazo[1,5-a]azepin-3-amine
• 9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-amine
• Epinastine base
• Wal 801
• (±)-Epinastine
• Epinastine

3-amino-9,13b-dihydro-1h-dibenz[c,f]imidazo[1,5-a]azepine

CAS: 80012-43-7

Formula: C₁₆H₁₅N₃

Purity: 98%

Color and Shape: Solid

Molecular weight: 249.3104

Ref: IN-DA00ID35

9,13B-Dihydro-1H-Dibenzo[c,f]Imidazo[1,5-A]Azepin-3-Amine

CAS: 80012-43-7

9,13B-Dihydro-1H-Dibenzo[c,f]Imidazo[1,5-A]Azepin-3-Amine

Purity: 98%

Molecular weight: 249.31g/mol

Ref: 54-OR1026295

Epinastine

CAS: 80012-43-7

Formula: C₁₆H₁₅N₃

Molecular weight: 249.31

Ref: 7W-GP7302

Epinastine

CAS: 80012-43-7

Formula: C₁₆H₁₅N₃

Purity: >98.0%(T)(HPLC)

Color and Shape: White to Light yellow powder to crystal

Molecular weight: 249.32

Ref: 3B-E1540

Epinastine

CAS: 80012-43-7

Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.

Formula: C₁₆H₁₅N₃

Purity: 99.94%

Color and Shape: Solid

Molecular weight: 249.31

Ref: TM-T60366