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CAS 80880-90-6

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Telenzepine

Description:
Telenzepine is a chemical compound classified as an anticholinergic agent, primarily used in the treatment of various gastrointestinal disorders. It functions by inhibiting the action of acetylcholine on muscarinic receptors, leading to reduced gastrointestinal motility and secretion. Telenzepine is known for its selective action, which minimizes side effects commonly associated with non-selective anticholinergics. The compound is typically administered in oral form and has been studied for its efficacy in managing conditions such as peptic ulcers and irritable bowel syndrome. Its pharmacokinetic profile indicates a relatively rapid absorption and a moderate half-life, allowing for effective therapeutic dosing. Additionally, Telenzepine's chemical structure features a unique arrangement that contributes to its pharmacological properties. As with many medications, potential side effects may include dry mouth, constipation, and blurred vision, which are typical of anticholinergic drugs. Overall, Telenzepine represents a valuable option in the pharmacotherapy of gastrointestinal disorders, with a focus on minimizing adverse effects while providing symptomatic relief.
Formula:C19H22N4O2S
InChI:InChI=1S/C19H22N4O2S/c1-13-18-14(12-26-13)19(25)20-15-5-3-4-6-16(15)23(18)17(24)11-22-9-7-21(2)8-10-22/h3-6,12H,7-11H2,1-2H3,(H,20,25)
InChI key:InChIKey=VSWPGAIWKHPTKX-UHFFFAOYSA-N
SMILES:C(CN1CCN(C)CC1)(=O)N2C=3C(C(=O)NC=4C2=CC=CC4)=CSC3C
Synonyms:
  • 10H-Thieno[3,4-b][1,5]benzodiazepin-10-one, 4,9-dihydro-3-methyl-4-[(4-methyl-1-piperazinyl)acetyl]-
  • 10H-thieno[3,4-b][1,5]benzodiazepin-10-one, 4,9-dihydro-3-methyl-4-[2-(4-methyl-1-piperazinyl)acetyl]-
  • 3-methyl-4-[(4-methylpiperazin-1-yl)acetyl]-4,9-dihydro-10H-thieno[3,4-b][1,5]benzodiazepin-10-one
  • 3-methyl-4-[(4-methylpiperazin-1-yl)acetyl]-4,9-dihydro-10H-thieno[3,4-b][1,5]benzodiazepin-10-one hydrochloride (1:1)
  • 4,9-Dihydro-3-methyl-4-[(4-methyl-1-piperazinylacetyl)]-10H-thieno[3,4-b][1,5]benzodiazepin-10-one
  • 4,9-Dihydro-3-methyl-4-[2-(4-methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-one
  • Telenzepine
  • (±)-Telenzepine
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