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CAS 82857-38-3

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Bopindolol malonate

Description:
Bopindolol malonate is a pharmaceutical compound primarily recognized for its role as a beta-blocker, which is used in the management of cardiovascular conditions such as hypertension and certain types of arrhythmias. It is characterized by its ability to selectively block beta-adrenergic receptors, leading to a decrease in heart rate and myocardial contractility. The malonate component indicates that it is a salt or ester derived from malonic acid, which may enhance its solubility and bioavailability. Bopindolol malonate exhibits a moderate lipophilicity, allowing it to penetrate biological membranes effectively. Its pharmacokinetic profile typically includes oral bioavailability, metabolism primarily in the liver, and renal excretion of metabolites. The compound is also noted for its potential side effects, which may include fatigue, dizziness, and gastrointestinal disturbances. As with other beta-blockers, caution is advised in patients with asthma or certain cardiovascular conditions. Overall, Bopindolol malonate represents a significant therapeutic option in the management of cardiovascular diseases.
Formula:C23H28N2O3·C3H4O4
InChI:InChI=1S/C23H28N2O3.C3H4O4/c1-16-13-19-20(25-16)11-8-12-21(19)27-15-18(14-24-23(2,3)4)28-22(26)17-9-6-5-7-10-17;4-2(5)1-3(6)7/h5-13,18,24-25H,14-15H2,1-4H3;1H2,(H,4,5)(H,6,7)
InChI key:InChIKey=LDOONRJGLKHGJI-UHFFFAOYSA-N
SMILES:O(CC(OC(=O)C1=CC=CC=C1)CNC(C)(C)C)C2=C3C(NC(C)=C3)=CC=C2.C(C(O)=O)C(O)=O
Synonyms:
  • Propanedioic acid, compd. with 2-[(1,1-dimethylethyl)amino]-1-[[(2-methyl-1H-indol-4-yl)oxy]methyl]ethyl benzoate (1:1)
  • 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), (+-)-, propanedioate (1:1) (salt)
  • 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), propanedioate (1:1) (salt)
  • LT 31-200
  • 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), propanedioate (1:1) (salt) (9CI)
  • 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), (±)-, propanedioate (1:1) (salt)
  • Propanedioic acid, compd. with 2-[(1,1-dimethylethyl)amino]-1-[[(2-methyl-1H-indol-4-yl)oxy]methyl]ethyl benzoate (1:1)
  • Wandonorm
  • Propanedioic acid, compd. with (+-)-2-[(1,1-dimethylethyl)amino]-1-[[(2-methyl-1H-indol-4-yl)oxy]methyl]ethyl benzoate (1:1)
  • Bopindolol hydrogen malonate
  • See more synonyms
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