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CAS 84370-95-6

:

clebopride maleate

Description:
Clebopride maleate is a pharmaceutical compound primarily used as an antiemetic and gastroprokinetic agent. It is a derivative of the substituted benzamide class and functions by antagonizing dopamine D2 receptors, which helps in alleviating nausea and vomiting. The maleate salt form enhances its solubility and stability, making it suitable for oral administration. Clebopride exhibits a moderate affinity for serotonin receptors, contributing to its therapeutic effects on gastrointestinal motility. The compound is typically administered in tablet form and is indicated for various gastrointestinal disorders, including functional dyspepsia and gastroparesis. Its pharmacokinetics involve absorption in the gastrointestinal tract, with metabolism primarily occurring in the liver. Side effects may include drowsiness, dry mouth, and gastrointestinal disturbances, which are common with many medications affecting the central nervous system. As with any medication, it is essential to use clebopride maleate under medical supervision to manage potential interactions and contraindications effectively.
Formula:C20H24ClN3O2.C4H4O4
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