CAS 851723-84-7

Timapiprant

CAS: 851723-84-7

Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).

Formula: C₂₁H₁₇FN₂O₂

Purity: 97.44% - 99.51%

Color and Shape: Solid

Molecular weight: 348.37

Ref: TM-T2664

Timapiprant

Controlled Product

CAS: 851723-84-7

Timapiprant is an amide that acts as a selective inhibitor of the prostanoid receptor CRTH2, which is involved in regulating the inflammatory response. Timapiprant inhibits skin eosinophilia, which is associated with inflammatory skin diseases such as atopic dermatitis and psoriasis. It has been shown to be safe in clinical trials and has a good safety profile. The drug's mechanism of action may be due to its ability to inhibit the production of IL-4 and IL-13 by Th2 cells and its ability to inhibit lung function. Timapiprant has shown efficacy in treating allergic rhinitis, asthma, chronic obstructive pulmonary disease, erythema multiforme, pyoderma gangrenosum, and other types of inflammatory skin diseases.

Formula: C₂₁H₁₇FN₂O₂

Purity: Min. 95%

Molecular weight: 348.37 g/mol

Ref: 3D-FF32729