CAS 85320-67-8

Ericolol

Description:

Ericolol, with the CAS number 85320-67-8, is a chemical compound that belongs to the class of beta-blockers, which are primarily used in the treatment of cardiovascular conditions. Characteristically, Ericolol exhibits selective antagonistic activity at beta-adrenergic receptors, particularly the beta-1 subtype, which makes it effective in managing hypertension and certain types of arrhythmias. The compound is known for its ability to reduce heart rate and myocardial contractility, thereby decreasing cardiac workload. Additionally, Ericolol may possess some intrinsic sympathomimetic activity, which can lead to a milder effect on heart rate compared to non-selective beta-blockers. Its pharmacokinetic profile typically includes oral bioavailability and a moderate half-life, allowing for once or twice-daily dosing. As with many beta-blockers, potential side effects may include fatigue, dizziness, and bradycardia. Overall, Ericolol represents a valuable therapeutic option in the management of cardiovascular diseases, although its specific clinical applications and efficacy should be evaluated in the context of individual patient needs and conditions.

Formula: C₁₈H₂₄ClNO₃

InChI: InChI=1S/C18H24ClNO3/c1-18(2,3)20-10-15(22)11-23-17-9-13(19)5-7-16(17)12-4-6-14(21)8-12/h5,7-9,15,20,22H,4,6,10-11H2,1-3H3

InChI key: InChIKey=QACGCDWSRFDWQO-UHFFFAOYSA-N

SMILES: O(CC(CNC(C)(C)C)O)C1=C(C=CC(Cl)=C1)C2=CC(=O)CC2

Synonyms:

• 3-[4-Chloro-2-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]phenyl]-2-cyclopenten-1-one
• Ericolol
• 2-Cyclopenten-1-one, 3-[4-chloro-2-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]phenyl]-, (±)-
• 2-Cyclopenten-1-one, 3-[4-chloro-2-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]phenyl]-

Ericolol

CAS: 85320-67-8

Ericolol is a beta blocker.

Formula: C₁₈H₂₄ClNO₃

Color and Shape: Solid

Molecular weight: 337.84

Ref: TM-T68552