CAS 85505-64-2

Vapiprost

Description:

Vapiprost, with the CAS number 85505-64-2, is a synthetic compound that belongs to the class of prostaglandin analogs. It is primarily studied for its potential therapeutic applications, particularly in the field of cardiovascular medicine. The substance exhibits vasodilatory properties, which means it can help widen blood vessels, thereby improving blood flow and reducing blood pressure. Vapiprost is known to interact with specific receptors in the body, influencing various physiological processes. Its chemical structure includes functional groups that contribute to its biological activity, making it a subject of interest in pharmacological research. While Vapiprost has shown promise in preclinical studies, further research is necessary to fully understand its efficacy, safety profile, and potential side effects in clinical settings. As with many compounds in this category, the development and application of Vapiprost are closely monitored to ensure compliance with regulatory standards and to optimize its therapeutic benefits.

Formula: C₃₀H₃₉NO₄

InChI: InChI=1S/C30H39NO4/c32-27-21-28(35-22-23-15-17-25(18-16-23)24-11-5-3-6-12-24)26(13-7-1-2-8-14-29(33)34)30(27)31-19-9-4-10-20-31/h1-3,5-6,11-12,15-18,26-28,30,32H,4,7-10,13-14,19-22H2,(H,33,34)/b2-1-/t26-,27-,28-,30+/m0/s1

InChI key: InChIKey=GQGRDYWMOPRROR-XUSMOFMBSA-N

SMILES: C(C/C=C\CCC(O)=O)[C@@H]1[C@H]([C@@H](O)C[C@@H]1OCC2=CC=C(C=C2)C3=CC=CC=C3)N4CCCCC4

Synonyms:

• (4E)-7-[(1R,2R,3S,5S)-5-(biphenyl-4-ylmethoxy)-3-hydroxy-2-piperidin-1-ylcyclopentyl]hept-4-enoic acid
• (4Z)-7-[(1R,2R,3S,5S)-5-([1,1′-Biphenyl]-4-ylmethoxy)-3-hydroxy-2-(1-piperidinyl)cyclopentyl]-4-heptenoic acid
• (4Z)-7-[(1R,2R,3S,5S)-5-(biphenyl-4-ylmethoxy)-3-hydroxy-2-piperidin-1-ylcyclopentyl]hept-4-enoic acid
• (4Z)-7-[(1R,2R,3S,5S)-5-(biphenyl-4-ylmethoxy)-3-hydroxy-2-piperidin-1-ylcyclopentyl]hept-4-enoic acid hydrochloride
• 4-Heptenoic acid, 7-(5-((1,1'-biphenyl)-4-ylmethoxy)-3-hydroxy-2-(1-piperidinyl)cyclopentyl)-, (1R-(1alpha(Z),2beta,3beta,5alpha))-
• 4-Heptenoic acid, 7-[(1R,2R,3S,5S)-5-([1,1′-biphenyl]-4-ylmethoxy)-3-hydroxy-2-(1-piperidinyl)cyclopentyl]-, (4Z)-
• 4-Heptenoic acid, 7-[5-([1,1′-biphenyl]-4-ylmethoxy)-3-hydroxy-2-(1-piperidinyl)cyclopentyl]-, [1R-[1α(Z),2β,3β,5α]]-
• Gr 32191
• Gr 322191
• Unii-H84Xt1Coau
• Vapiprost [INN:BAN]
• Vapiprostum
• Vapiprostum [Latin]

Vapiprost

CAS: 85505-64-2

Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.

Formula: C₃₀H₃₉NO₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 477.64

Ref: TM-T24931

Vapiprost

CAS: 85505-64-2

Vapiprost is a peptide inhibitor of the calmodulin-dependent protein kinase II. This enzyme phosphorylates the amino acid residue Thr-286 in the regulatory domain of the protein phosphatase 2A, which causes it to dephosphorylate and activate its substrates. Vapiprost prevents this phosphorylation and activation, thus inhibiting PKII activity. It is not active against other kinases or phosphatases.

Formula: C₃₀H₃₉NO₄

Purity: Min. 95%

Molecular weight: 477.60 g/mol

Ref: 3D-KDA50564