CAS 86880-51-5

Epanolol

Description:

Epanolol, identified by its CAS number 86880-51-5, is a beta-adrenergic antagonist, commonly referred to as a beta-blocker. This class of compounds is primarily used in the management of cardiovascular conditions, including hypertension and arrhythmias. Epanolol exhibits selectivity for beta-1 adrenergic receptors, which are predominantly found in the heart, leading to a decrease in heart rate and myocardial contractility. The compound is characterized by its ability to reduce cardiac output and lower blood pressure, making it effective in treating various heart-related ailments. Additionally, beta-blockers like Epanolol may have applications in anxiety management and migraine prophylaxis due to their effects on the sympathetic nervous system. The pharmacokinetics of Epanolol involve oral administration, with absorption and metabolism occurring in the liver. As with other beta-blockers, potential side effects may include fatigue, dizziness, and bradycardia. It is essential for patients to consult healthcare professionals before starting treatment with Epanolol to ensure it is appropriate for their specific health conditions.

Formula: C₂₀H₂₃N₃O₄

InChI: InChI=1/C20H23N3O4/c21-12-16-3-1-2-4-19(16)27-14-18(25)13-22-9-10-23-20(26)11-15-5-7-17(24)8-6-15/h1-8,18,22,24-25H,9-11,13-14H2,(H,23,26)

InChI key: InChIKey=YARKMNAWFIMDKV-UHFFFAOYSA-N

SMILES: O(CC(CNCCNC(CC1=CC=C(O)C=C1)=O)O)C2=C(C#N)C=CC=C2

Synonyms:

• (+-)-N-(2-((3-(o-Cyanophenoxy)-2-hydroxypropyl)amino)ethyl)-2-(p-hydroxyphenyl)acetamide
• Benzeneacetamide, N-(2-((3-(2-cyanophenoxy)-2-hydroxypropyl)amino)ethyl)-4-hydroxy-
• Epanolol [INN:BAN]
• Epanololum
• Epanololum [Latin]
• Ici 141292
• N-(2-{[3-(2-cyanophenoxy)-2-hydroxypropyl]amino}ethyl)-2-(4-hydroxyphenyl)acetamide
• N-[2-[[3-(2-Cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-4-hydroxybenzeneacetamide
• Unii-9Kgc55Kp6A
• Visacor
• Epanolol

Epanolol

Controlled Product

CAS: 86880-51-5

Formula: C₂₀H₂₃N₃O₄

Color and Shape: Neat

Molecular weight: 369.414

Ref: TR-E565500

Epanolol

CAS: 86880-51-5

Epanolol is a beta-adrenergic receptor antagonist that is used to treat heart failure, high blood pressure, and other cardiovascular diseases. It has been shown to increase urine production by reducing the concentration of natriuretic peptides in the body. Epanolol also has anti-inflammatory effects and can be used for the treatment of skin conditions such as psoriasis. Epanolol has a terminal half-life of about six hours and an effective dose range of 10-40 mg/day.

Formula: C₂₀H₂₃N₃O₄

Purity: Min. 95%

Molecular weight: 369.4 g/mol

Ref: 3D-LDA88051

Epanolol

CAS: 86880-51-5

Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.

Formula: C₂₀H₂₃N₃O₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 369.41

Ref: TM-T11608