CAS 879497-82-2

L-Valine, L-a-aspartyl-3-mercapto-L-valyl-L-phenylalanyl-D-tryptophyl-(2S)-2,4-diaminobutanoyl-L-tyrosyl-L-cysteinyl-,cyclic (2®7)-disulfide

Description:

L-Valine, L-a-aspartyl-3-mercapto-L-valyl-L-phenylalanyl-D-tryptophyl-(2S)-2,4-diaminobutanoyl-L-tyrosyl-L-cysteinyl-, cyclic (2®7)-disulfide, identified by CAS number 879497-82-2, is a complex peptide with a unique cyclic disulfide structure. This compound features a sequence of amino acids that includes valine, aspartic acid, phenylalanine, tryptophan, tyrosine, and cysteine, which contribute to its biological activity and structural stability. The presence of the cyclic disulfide linkage enhances its resistance to enzymatic degradation, making it potentially useful in pharmaceutical applications. The mercapto group indicates the presence of a thiol, which can participate in redox reactions and may play a role in biological signaling pathways. Overall, this compound's intricate structure suggests it may have specific interactions with biological targets, warranting further investigation into its potential therapeutic uses and mechanisms of action.

Formula: C₅₀H₆₄N₁₀O₁₂S₂

Synonyms:

• Ufp803

UFP-803

CAS: 879497-82-2

UT receptor ligand acts mainly as silent antagonist with slight agonist effects; blocks U-II in rat aorta, pIC50 = 7.46, & inhibits plasma leakage in mice.

Formula: C₅₀H₆₄N₁₀O₁₂S₂

Purity: 98%

Color and Shape: Solid

Molecular weight: 1061.24

Ref: TM-TP2104

UFP 803

CAS: 879497-82-2

UFP 803 is a ligand for the urotensin-II receptor. It has been shown to have effects on the release of neurotransmitters, such as noradrenaline, serotonin, and dopamine. In vivo assays show that UFP 803 inhibits the excitatory effect of glutamate on neuronal activity in the brain by blocking the release of neurotransmitters from neurons. This drug also reduces inflammation and prevents extravasation in animal models. UFP 803 acts by binding with high affinity to urotensin II receptors and inhibiting cellular proliferation induced by urotensin-II.

Formula: C₅₀H₆₄N₁₀O₁₂S₂

Purity: Min. 95%

Molecular weight: 1,061.2 g/mol

Ref: 3D-EKB49782