CAS 88373-72-2

(D-pen2,pen5)-enkephalin

Description:

(D-pen2,pen5)-enkephalin, also known as a synthetic peptide, is a member of the enkephalin family, which are endogenous opioid peptides that play a crucial role in pain modulation and neurotransmission. This compound is characterized by its specific amino acid sequence, which includes two D-phenylalanine residues at positions 2 and 5, contributing to its stability and affinity for opioid receptors. It exhibits potent analgesic properties and acts primarily on the delta-opioid receptors, influencing pain perception and emotional responses. The structure of (D-pen2,pen5)-enkephalin allows it to mimic the natural enkephalins, making it a valuable compound in pharmacological research. Its stability against enzymatic degradation enhances its potential therapeutic applications. Additionally, this peptide is often studied for its effects on the central nervous system and its potential use in treating conditions such as chronic pain and addiction. Overall, (D-pen2,pen5)-enkephalin represents a significant interest in the field of medicinal chemistry and neuropharmacology.

Formula: C₃₀H₃₉N₅O₇S₂

Synonyms:

• H-Tyr-D-Pen-Gly-Phe-Pen-OH (Disulfide bond)