CAS 89197-32-0

Efaroxan

Description:

Efaroxan is a chemical compound classified as an atypical antipsychotic and is primarily known for its role as a selective antagonist of the α2-adrenergic receptor. It has been studied for its potential therapeutic effects in treating various psychiatric disorders, particularly in enhancing cognitive function and alleviating symptoms of depression. Efaroxan exhibits a unique mechanism of action by modulating neurotransmitter systems, particularly norepinephrine and serotonin, which are crucial in mood regulation and cognitive processes. The compound is characterized by its ability to cross the blood-brain barrier, allowing it to exert effects on the central nervous system. Additionally, Efaroxan has been investigated for its potential neuroprotective properties and its influence on metabolic processes. Its pharmacokinetics, including absorption, distribution, metabolism, and excretion, are essential for understanding its efficacy and safety profile in clinical applications. As research continues, Efaroxan may offer insights into novel treatment strategies for mental health disorders.

Formula: C₁₃H₁₆N₂O

InChI: InChI=1S/C13H16N2O/c1-2-13(12-14-7-8-15-12)9-10-5-3-4-6-11(10)16-13/h3-6H,2,7-9H2,1H3,(H,14,15)

InChI key: InChIKey=RATZLMXRALDSJW-UHFFFAOYSA-N

SMILES: C(C)C1(CC=2C(O1)=CC=CC2)C=3NCCN3

Synonyms:

• (+-)-2-(2-Ethyl-2,3-dihydro-2-benzofuranyl)-2-imidazoline
• 1H-Imidazole, 2-(2-ethyl-2,3-dihydro-2-benzofuranyl)-4,5-dihydro-
• 2-(2-Ethyl-2,3-dihydro-2-benzofuranyl)-4,5-dihydro-1H-imidazole
• 2-(2-ethyl-2,3-dihydro-1-benzofuran-2-yl)-4,5-dihydro-1H-imidazole
• 2-(2-ethyl-2,3-dihydro-1-benzofuran-2-yl)-4,5-dihydro-1H-imidazole hydrochloride (1:1)
• Efaroxan [INN:BAN]
• Efaroxano
• Efaroxano [INN-Spanish]
• Efaroxanum
• Efaroxanum [INN-Latin]
• Unii-G00490L21H