CAS 911-65-9

Etonitazene

Description:

Etonitazene is a synthetic opioid that belongs to the class of compounds known as benzimidazole derivatives. It is characterized by its potent analgesic properties, which are significantly stronger than those of morphine. Etonitazene acts primarily on the mu-opioid receptors in the central nervous system, leading to effects such as pain relief, sedation, and euphoria. Its chemical structure includes a nitrogen-containing heterocyclic ring, contributing to its pharmacological activity. Due to its high potency, Etonitazene poses a considerable risk for respiratory depression and overdose, similar to other opioids. It is classified as a controlled substance in many jurisdictions due to its potential for abuse and addiction. Additionally, research on Etonitazene is limited, and its safety profile is not well-established, making it a substance of concern in the context of public health and drug regulation. As with all opioids, caution is advised in its use, and it should only be administered under strict medical supervision.

Formula: C₂₂H₂₈N₄O₃

InChI: InChI=1S/C22H28N4O3/c1-4-24(5-2)13-14-25-21-12-9-18(26(27)28)16-20(21)23-22(25)15-17-7-10-19(11-8-17)29-6-3/h7-12,16H,4-6,13-15H2,1-3H3

InChI key: InChIKey=PXDBZSCGSQSKST-UHFFFAOYSA-N

SMILES: C(CN(CC)CC)N1C=2C(N=C1CC3=CC=C(OCC)C=C3)=CC(N(=O)=O)=CC2

Synonyms:

• 1-(2-Diethylaminoethyl)-2-(4-Ethoxybenzyl)-5-Nitrobenzimidazole
• 1-(2-Diethylaminoethyl)-2-p-ethoxybenzyl-5-nitrobenzimidazole
• 1-(β-Diethylaminoethyl)-2-(p-ethoxybenzyl)-5-nitrobenzimidazole
• 1H-Benzimidazole-1-ethanamine, 2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-5-nitro-
• 2-[(4-Ethoxyphenyl)methyl]-N,N-diethyl-5-nitro-1H-benzimidazole-1-ethanamine
• 2-[2-(4-ethoxybenzyl)-5-nitro-1H-benzimidazol-1-yl]-N,N-diethylethanamine
• Arc 1G2
• Ba 20684
• Benzimidazole, 1-[2-(diethylamino)ethyl]-2-(p-ethoxybenzyl)-5-nitro-
• Ciba 20-684BA
• Etobedolum
• Etonitazine
• N-[2-[2-(4-Ethoxybenzyl)-5-nitrobenzimidazol-1-yl]ethyl]diethylamine

Etonitazene

Controlled Product

CAS: 911-65-9

Applications Etonitazene is a μ-opioid receptor agonist structurally related to Clonitazene (C587135).
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References May, T., et al.: Neurosci. Lett., 275, 109 (1999); Piepponen, T.P., et al.: Pharmacol. Biochem. Behav., 63, 245 (1999); Baumgartner, A., et al.: Psychopharmacology, 135, 63 (1998)

Formula: C₂₂H₂₈N₄O₃

Color and Shape: Neat

Molecular weight: 396.48

Ref: TR-E933600

Etonitazene-d5

Controlled Product

CAS: 911-65-9

Applications Etonitazene-d5 is the isotope labelled analog of Etonitazene (E933600); a μ-opioid receptor agonist structurally related to Clonitazene (C587135).
References May, T., et al.: Neurosci. Lett., 275, 109 (1999); Piepponen, T.P., et al.: Pharmacol. Biochem. Behav., 63, 245 (1999); Baumgartner, A., et al.: Psychopharmacology, 135, 63 (1998)

Formula: C₂₂D₅H₂₃N₄O₃

Color and Shape: Light Yellow

Molecular weight: 401.51

Ref: TR-E933602