CAS 923270-50-2

Cyclopenta[c]pyrrole-1-carboxaMide, (2S)-2-cyclohexyl-N-(2-pyrazinylcarbonyl)glycyl-3-Methyl-L-valyl-N-[(1R)-1-[2-(cyclopropylaMino)-2-oxoacetyl]butyl]octahydro-, (1S,3aR,6aS)-

Description:

Cyclopenta[c]pyrrole-1-carboxamide, with the CAS number 923270-50-2, is a complex organic compound characterized by its unique bicyclic structure that includes a cyclopentane and pyrrole moiety. This compound features multiple functional groups, including an amide and various substituents that contribute to its chemical reactivity and potential biological activity. The presence of a cyclohexyl group and a pyrazinylcarbonyl moiety suggests that it may exhibit interesting interactions in biological systems, possibly influencing its pharmacological properties. Additionally, the stereochemistry indicated by the (2S) and (1R) designations suggests that the compound has specific spatial arrangements that could affect its binding affinity and selectivity for biological targets. Overall, the structural complexity and functional diversity of this compound make it a subject of interest in medicinal chemistry and drug development, particularly in the context of exploring new therapeutic agents.

Formula: C₃₆H₅₃N₇O₆

Synonyms:

• Telaprevir (R)-Isomer
• Cyclopenta[c]pyrrole-1-carboxaMide, (2S)-2-cyclohexyl-N-(2-pyrazinylcarbonyl)glycyl-3-Methyl-L-valyl-N-[(1R)-1-[2-(cyclopropylaMino)-2-oxoacetyl]butyl]octahydro-, (1S,3aR,6aS)-
• (R)-Telaprevir
• (1S,3aR,6aS)-(2S)-2-Cyclohexyl-N-(2-pyrazinylcarbonyl)glycyl-3-methyl-L-valyl-N-[(1R)-1-[2-(cyclopropylamino)-2-oxoacetyl]butyl]octahydrocyclopenta[c]pyrrole-1-carboxamide

Cyclopenta[c]pyrrole-1-carboxaMide, (2S)-2-cyclohexyl-N-(2-pyrazinylcarbonyl)glycyl-3-Methyl-L-valyl-N-[(1R)-1-[2-(cyclopropylaMino)-2-oxoacetyl]butyl]octahydro-, (1S,3aR,6aS)-

CAS: 923270-50-2

Formula: C₃₆H₅₃N₇O₆

Purity: 97%

Molecular weight: 679.8493

Ref: IN-DA00GWLU

(R)-Telaprevir-d4

Controlled Product

CAS: 923270-50-2

Applications (R)-Telaprevir-d4 is the labeled analog of (R)-Telaprevir, an enantiomer of Telaprevir (T015650). Telaprevir is an known inhibitor of the hepatitis C virus NS3-4A protease. It is a COVID19-related research product.
References Francois, J., et al.: J. Medn. Chem., 52. 7993 (2009); Kieffer, T., et al.: Hepatology, 46, 631 (2007), Zhou, Y., et al.: Antimicrob. Agents Chemother., 52, 110 (2008), Hezode, C., et al.: N. Engl. J. Med., 360, 1839 (2009);

Formula: C₃₆H₄₉D₄N₇O₆

Color and Shape: Neat

Molecular weight: 683.87

Ref: TR-T015662

(R)-Telaprevir

Controlled Product

CAS: 923270-50-2

Applications (R)-Telaprevir is an enantiomer of Telaprevir (T015650), an inhibitor of the hepatitis C virus NS3-4A protease. It is a COVID19-related research product.
References Francois, J., et al.: J. Medn. Chem., 52. 7993 (2009); Kieffer, T., et al.: Hepatology, 46, 631 (2007), Zhou, Y., et al.: Antimicrob. Agents Chemother., 52, 110 (2008), Hezode, C., et al.: N. Engl. J. Med., 360, 1839 (2009);

Formula: C₃₆H₅₃N₇O₆

Color and Shape: Neat

Molecular weight: 679.85

Ref: TR-T015660

(R)-Telaprevir

CAS: 923270-50-2

Telaprevir is a small molecule that binds to the cytoplasmic domain of the human immunodeficiency virus type 1 (HIV-1) envelope protein, blocking its fusion with host cells. Telaprevir is also an inhibitor of hepatitis C virus (HCV) NS3 protease. The binding of telaprevir to HIV-1 and HCV is selective and reversible. This drug has been shown to be effective in inhibiting the replication of HIV-1 and HCV in vitro, as well as in clinical trials. Telaprevir binds to the active site of the protease, preventing cleavage of a polyprotein into three parts: p7, p2, and p6. Telaprevir is an ion channel blocker that inhibits potassium channels. It can be used as a research tool for studying ligand-receptor interactions or protein interactions with peptides. Telaprevir is a high purity product with CAS No.

Formula: C₃₆H₅₃N₇O₆

Purity: Min. 95%

Molecular weight: 679.8 g/mol

Ref: 3D-YLB27050